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4-[(4-fluorophenyl)methyl]-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]piperazine-1-carboxamide
1-(adamantan-1-yl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
6-{[ethyl(methyl)amino]methyl}-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
N-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
5-methyl-4-[4-(pyridin-3-yl)piperazin-1-yl]pyrimidin-2-amine
2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]pyridine-4-carboxamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-cyclopropylpropanamide
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-methylpropanamide
1-(pyrrolidin-1-yl)-2-{4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazin-1-yl}ethan-1-one
5-(benzylamino)-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{4-[4-(4-ethylpiperazin-1-yl)piperidine-1-carbonyl]piperidin-1-yl}-4-methyl-6-(propan-2-yl)quinazoline
7-(1,3-benzothiazol-2-yl)-4-{[4-(methylsulfanyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,4S)-1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(morpholin-4-yl)pyrrolidin-3-ol
5-{[2-(pyrrolidin-1-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
1-methyl-3-propyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide
8-fluoro-2-{[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}quinolin-4-ol
N,2-dimethyl-3-(morpholin-4-yl)-N-(quinolin-6-ylmethyl)propanamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(thiophen-3-ylmethyl)piperazine
1-({3-[4-(morpholin-4-yl)butoxy]phenyl}methyl)-1,4-diazepan-5-one
4-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-N-(propan-2-yl)pyridine-2-carboxamide
2-(cyclohex-1-en-1-yl)-1-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
(1S,5R)-3-[3-(4-ethyl-5-hydroxy-3-methyl-1H-pyrazol-1-yl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[3-methyl-7-(1-methylpiperidine-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
4-{[methyl(prop-2-en-1-yl)amino]methyl}-N-(2,4,6-trimethylpyridin-3-yl)benzamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-oxo-2-[2-(piperidin-1-yl)ethyl]-2,3-dihydro-1H-isoindole-5-carboxamide
(1S,5R)-3-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
6-oxo-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)pyridine-3-carboxylic acid
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(2-methoxyphenyl)propyl]propanamide
1-[(4-fluorophenyl)methyl]-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
2-ethyl-8-(4-phenoxybutanoyl)-2,8-diazaspiro[4.5]decan-3-one
N-(1-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
2-methoxy-N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-{2-[1-(1H-indazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-{3-[methyl(phenyl)amino]propyl}-1-(pyrimidin-2-yl)piperidin-4-amine
3-benzyl-1-(3-methoxypropyl)-8-{[3-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}acetamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(4-hydroxy-4-phenylpiperidin-1-yl)-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
N-(3-hydroxy-3-phenylpropyl)-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
5-(oxolan-2-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]thiophene-2-carboxamide
3-(2-methoxyethyl)-5-(2-phenylethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-[5-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)thiophen-2-yl]acetamide
5-[1-(5-methoxy-1H-indole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-benzyl-9-(piperidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-chloro-4-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
(3aR,5R,6S,7aS)-2-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-octahydro-1H-isoindole-5,6-diol
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[3-(morpholin-4-yl)propyl]-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
8-(1-methyl-1H-pyrazole-5-carbonyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one