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4-{2-[2-(2-chloro-3,4-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}pyridine
N-[(1-ethylpyrrolidin-2-yl)methyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
2-(1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
4-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl]benzoic acid
(1-{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-yl)methanol
N-[(3-ethoxyphenyl)methyl]-N-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}cyclopropanamine
5-(furan-2-yl)-3-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
4-(3-{[1-(ethanesulfonyl)piperidin-4-yl]oxy}benzoyl)morpholine
3-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
3-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
3-hydroxy-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-2,7-dimethyl-N-(prop-2-en-1-yl)quinoline-4-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-cyclopentyl-4-({[(2-fluoro-4,5-dimethoxyphenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
1-[(2-chlorophenyl)methyl]-4-[(cyclopropylmethyl)amino]pyrrolidin-2-one
3,5-difluoro-2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2,8-dimethyl-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}quinoline
1-methyl-4-[2-(2-phenylphenyl)-1H-imidazol-1-yl]piperidine
6-cyclobutanecarbonyl-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-(3-{[(4-chlorophenyl)methyl]sulfanyl}propyl)-1,5-dimethyl-1H-pyrazole-4-carboxamide
1-[3-(2-phenylethyl)piperidine-1-carbonyl]cyclobutan-1-amine
1-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
4-ethyl-3-{1-[2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,7aR)-1-(4-methylpent-3-en-1-yl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5,6,7,8-tetrahydroquinazolin-2-amine
(1R,5R)-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
3-(2-chlorobenzoyl)-N-[(3-fluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-({5-[(2-fluoro-5-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(morpholin-3-yl)ethan-1-one
5-[1-(2-methoxybenzoyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
4-benzyl-1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-1,4-diazepan-5-one
6-methyl-2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
N,N-dimethyl-3-{1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidin-3-yl}propanamide
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-2-propyl-1,3-thiazole-4-carboxamide
5-(3-tert-butyl-5-methylphenyl)pyrazine-2-carboxylic acid
2-methoxy-5-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}phenol
8-fluoro-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}quinoline-2-carboxamide
5-butyl-4-methyl-6-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]pyrimidin-2-amine
4-[4-(cyclohex-3-en-1-ylmethyl)piperazin-1-yl]-2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(aminomethyl)-4-[2-(4-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
9-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(methylsulfanyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N,5-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[3-(pyridin-3-yl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
N-[2-(dimethylamino)ethyl]-3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}propanamide
3-[1-(2-methoxyacetyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
3-(2-chlorophenoxy)-1-(7-methyl-1-benzofuran-2-carbonyl)azetidine
2-{4-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]quinazolin-2-yl}ethan-1-amine