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5-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2-methylpyridine
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N,2-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-(2,6-dimethoxypyridin-3-yl)-2-{methyl[2-(pyrrolidin-1-yl)ethyl]amino}acetic acid
(1S,5R)-3-(pyrazin-2-yl)-6-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
ethyl 3-[(3-chlorophenyl)methyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-3-carboxylate
3-(3-chlorobenzoyl)-1-(2-methoxy-5-methylbenzenesulfonyl)piperidine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-(2-methyl-1H-indol-1-yl)propanamide
4-[7-(3-ethyl-1H-pyrazole-5-carbonyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
5-(1-aminocyclopropanecarbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-methoxy-9-[2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecane
(3aR,7aS)-2-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
methyl 6-{[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]methyl}pyridine-2-carboxylate
N-[2-(dimethylamino)ethyl]-3-{1-[2-(furan-2-yl)-2-oxoacetyl]piperidin-4-yl}propanamide
(4-{3-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}phenyl)methanol
1-(1,3-benzothiazol-2-yl)-N-[1-(furan-2-ylmethyl)piperidin-4-yl]piperidin-3-amine
ethyl 2-({5-[2-amino-3-cyano-6-(propan-2-yl)pyridin-4-yl]pyrimidin-2-yl}amino)acetate
8-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
(1R,5R)-3-cyclobutanecarbonyl-6-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[1-(3-fluoropropyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}adamantane-1-carboxamide
1-(4-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
5-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(methylsulfanyl)pyrimidine
1-[(4,5-dimethylfuran-2-yl)methyl]-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
3-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-6-(trifluoromethyl)pyridin-2-ol
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-1-methylazepane-2-carboxamide
11-{[(3,4-difluorophenyl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3S,9aR)-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2-methyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(3-fluorophenyl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}propan-1-one
1-phenyl-4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazin-2-one
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
1-methyl-3-[1-(morpholine-3-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[3-(pyrrolidine-1-sulfonyl)thiophene-2-carbonyl]piperazine-2-carboxylic acid
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamide
N-{4-methyl-2-[2-(2-oxopyrrolidin-1-yl)propanamido]phenyl}cyclohexanecarboxamide
1-[(6-methylpyridin-2-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-cyclopentyl-1-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-[(3-chlorophenyl)methyl]-5-{2-[(pyridin-2-ylmethyl)amino]ethyl}pyrrolidin-2-one
6-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
(3S,4R)-4-(2-methylphenyl)-1-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)pyrrolidine-3-carboxylic acid
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)oxolane-2-carboxamide
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidin-2-amine
1-[(4-methylphenyl)methyl]-5-oxo-N-[2-(1H-pyrrol-1-yl)ethyl]pyrrolidine-3-carboxamide
1-methyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-(5-propylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)acetamide
N-[2-(4-chlorobenzenesulfonamido)ethyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
(4aR,7aS)-1-acetyl-4-[(3-hydroxy-4-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione