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(2S,4S)-N,N-diethyl-1-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]pyrrolidine-2-carboxamide
6-(aminomethyl)-N-[(3-chloro-2,6-difluorophenyl)methyl]pyrimidin-4-amine
1-[(2-cyanophenyl)methyl]-3-propylpiperidine-3-carboxylic acid
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyridine
methyl 1-{4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxybenzoyl}piperidine-2-carboxylate
1-[3-(furan-2-yl)-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-1-methanesulfonyl-4-[(trimethyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,5S)-N3-(4-fluorophenyl)-N5-(2-phenylethyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
[3-(4-ethylphenyl)propyl](methyl)(pyridin-3-ylmethyl)amine
5-(morpholin-4-ylmethyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]furan-3-carboxamide
(4R)-N,3-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazolidine-4-carboxamide
N-(2,3-dihydro-1-benzofuran-3-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
6-[(diethylamino)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(2S,4S)-1-(2,2-diphenylethyl)-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
1-{4-[4-(pyridin-4-yl)piperazine-1-carbonyl]thiophen-2-yl}ethan-1-one
{2-fluoro-5-[5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]phenyl}methanol
(3aS,6aS)-2-[3-(dimethylamino)benzoyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-4-{[(5-methyl-1,3,4-oxadiazol-2-yl)amino]methyl}-1,2,3,4-tetrahydroquinolin-2-one
N-[(2S,4R,6S)-2-benzyl-6-(4-oxo-4H-chromen-3-yl)oxan-4-yl]acetamide
4-phenyl-5-[2-(prop-2-yn-1-yloxy)phenyl]-1-(pyrrolidin-3-yl)-1H-imidazole
6-(5-methyl-2-{[2-(morpholin-4-yl)propanamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxamide
N-ethyl-4-hydroxy-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
{1-[(2,3,4-trifluorophenyl)methyl]azepan-2-yl}methanol
(1R,7S)-3-cycloheptyl-N-methyl-4-oxo-N-(pyrazin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[4-({4-[5-(3-fluorophenyl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenyl]acetamide
(3aS,6aS)-2-(dimethylsulfamoyl)-5-(pyrimidin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(2-fluorophenyl)methyl]-6-oxo-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
5-ethyl-6-methyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
1-ethyl-N,5-dimethyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(2-methyloxolan-2-yl)-1H-1,2,4-triazole
N,2-dimethyl-N-(quinolin-5-ylmethyl)oxane-2-carboxamide
1-[2-(2,5-dimethoxybenzenesulfonamido)ethyl]-N-phenyl-1H-1,2,3-triazole-4-carboxamide
2-{1-[(5-methylfuran-2-yl)methyl]-4-(thian-4-yl)piperazin-2-yl}ethan-1-ol
1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-phenylazepane
3-(4-chloro-1H-pyrazol-1-yl)-N-[(4-methoxyphenyl)methyl]-N-propylpropanamide
1-(2-amino-6-methylpyrimidin-4-yl)-4-(3-tert-butyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2S,3R)-2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-hydroxybutanamide
3-{1-[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]piperidin-2-yl}pyridine
3-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}azetidin-3-yl)pyridine
1-(difluoromethyl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-pyrazole-3-carboxamide
3-{2-[(4aS,8aS)-7-ethyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
1,5-dimethyl-3-{[2-(thiophen-3-yl)-1H-imidazol-1-yl]methyl}-1H-indazole
N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-4-[(3-methylpiperidin-1-yl)methyl]benzamide
(1s,4s)-4-{4-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(2-{2-[2-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}ethyl)-4H-1,2,4-triazole
[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl][(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine