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1-(1-{2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
N-[(5-chlorothiophen-2-yl)methyl]-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(3S,4R)-1-[2-(2-fluorophenyl)benzoyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[3-(morpholin-4-yl)propyl]piperidine-3,5-dicarboxamide
1-(5-acetyl-2-ethoxyphenyl)-3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethylurea
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[2-(ethylamino)pyrimidin-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
4-(6-chloroquinolin-2-yl)-1-methylpiperazin-2-one
1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)cyclobutanecarboxamide
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-ethyl-2,5-dihydro-1H-pyrrole-1-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-[(3-methoxyphenyl)amino]butanamide
5-(4-methylphenyl)-4-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-3-yl}pyrimidine
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}cyclohexanecarboxamide
1-{imidazo[1,2-b]pyridazin-6-yl}-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazine
1-methyl-8-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-methyl-5-[(6-oxo-5,6-dihydrophenanthridin-5-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-5-methyl-1,2-oxazole-4-carboxamide
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
(1S,6R)-3-(3-chloro-4-propoxybenzoyl)-3,9-diazabicyclo[4.2.1]nonane
N,N-dimethyl-2-{[2-(methylsulfanyl)acetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)pyrimidine
4-[(5-{[(2-chloro-5-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-(2,2-dimethyloxan-4-yl)-5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-N-(2-fluorophenyl)propanamide
{1-[7-(thiophene-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-yl}methanol
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
1-methyl-1'-(5-propyl-1,2-oxazole-3-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-[3-(1H-pyrazol-4-yl)benzoyl]morpholine
4-amino-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)butan-1-one
N-[(4-{3,9-diazaspiro[5.5]undecane-3-carbonyl}phenyl)methyl]-2-methylpropanamide
5-fluoro-2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
2-amino-4-cyclopropyl-6-(5-methylfuran-2-yl)pyridine-3-carbonitrile
4-[(2-hydroxyphenyl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4S)-N-ethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetamido]-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
(4aR,7aS)-1-acetyl-4-[2-(1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methoxy-N-{2-[(2R)-5-oxopyrrolidine-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}benzamide
N-({6-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridin-3-yl}methyl)acetamide
3-({methyl[(2-methylpyridin-4-yl)methyl]amino}methyl)benzoic acid
N-[3-(methylamino)propyl]-N'-(2-methylphenyl)propanediamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
N-[(4-methoxyphenyl)methyl]-1-methyl-N-propyl-1H-indazole-3-carboxamide
1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxylic acid
2-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-6-fluorophenol
N,N-diethyl-1-(5-methyl-1,3-oxazole-4-carbonyl)pyrrolidin-3-amine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-3-acetamidobenzamide
(2R,3R)-3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-[2-(2,6-dimethoxyphenoxy)ethyl]-5,6-dihydro-1,6-naphthyridin-5-one