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N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
2-methoxy-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyridine-4-carboxamide
(3aR,6aR)-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
methyl({[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
4-cyclopropanecarbonyl-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N,N-dimethyl-5-({3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}methyl)furan-2-carboxamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-cyclopentanecarbonyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-4-carboxamide
3-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
N-methyl-3-(3-methylpiperidin-1-yl)-N-[(3-methylthiophen-2-yl)methyl]propanamide
3-{3-[cyclohexyl(methyl)amino]propyl}-8-[(3-methylpyridin-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-4-(2-phenylethyl)piperazine
N-[(3R,4S)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]ethane-1-sulfonamide
N-(furan-2-ylmethyl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}propanamide
(4aS,8aR)-1-(2-aminoethyl)-6-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-decahydro-1,6-naphthyridin-2-one
N-{1-oxaspiro[4.4]nonan-3-yl}-2-(5-phenyl-4H-1,2,4-triazol-3-yl)acetamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
2-ethyl-9-(1,3-thiazol-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-hydroxy-4-(methylsulfanyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}butanamide
(4aS,7aR)-1-[(3,5-dichlorophenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{3-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
6-[4-(2-methylphenoxy)piperidin-1-yl]pyrimidine-2,4-diamine
4-[(3-phenylpiperidin-1-yl)methyl]-1H-pyrazole-3-carboxylic acid
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
5-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
2-ethoxy-1-[6-hydroxy-4-(quinolin-6-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
2-(4-chlorophenyl)-4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}morpholine
methyl 3-(cyclobutylmethoxy)-5-[methyl(oxan-4-yl)carbamoyl]benzoate
ethyl 4-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]piperazine-1-carboxylate
1-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-phenylpiperidin-4-yl)ethan-1-one
2-[9-(2-ethylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2-methoxy-5-methylbenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
3-{[(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
1-{pyrazolo[1,5-a]pyridine-3-carbonyl}azepan-4-amine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(4-methoxyphenyl)-4-methyl-1H-pyrazol-1-yl]acetamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[3-(pyridin-4-yl)azetidin-1-yl]propan-1-one
1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-4-(thiophen-2-ylmethyl)piperazine
1-[(3-methylphenyl)methyl]-4-(2-propylpyridine-4-carbonyl)piperazine
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(2-propoxyethyl)-1,4-diazepane
4-({[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]carbamoyl}amino)-N,N-diethyl-3-methylbenzamide
N-methyl-5-(phenoxymethyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-3-carboxamide
N-[(2S,4R,6S)-2-benzyl-6-[2-(pyridin-2-yl)pyrimidin-5-yl]oxan-4-yl]acetamide
2-[4-(propan-2-yl)morpholin-2-yl]-1-[3-(pyridin-4-yl)azetidin-1-yl]ethan-1-one
1-[(3,4-dichlorophenyl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
1-[(4-methoxyphenyl)methyl]-4-(4-propylbenzoyl)piperazin-2-one
2-ethyl-7-methoxy-4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-N-(propan-2-yl)pyrimidin-2-amine