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N-(3-methyl-1,2,4-thiadiazol-5-yl)-5-(1-propylpyrrolidin-2-yl)thiophene-2-carboxamide
2-({1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}amino)pyridine-3-carbonitrile
4-acetyl-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
(3S,4S)-1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-4-propylpyrrolidine-3-carboxylic acid
3,4,7-trimethyl-N,N-bis(1,3-oxazol-4-ylmethyl)-1H-indole-2-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-4-(pyridin-3-yl)pyrimidin-2-amine
4-chloro-N-[(4,6-dimethylpyridin-2-yl)methyl]-N,1-dimethyl-1H-pyrazole-5-carboxamide
N-(pyridin-2-ylmethyl)-1-[1-(pyrimidin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
6-cyclopropyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrimidin-4-amine
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
1-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
5-[4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-N-(4-methylpyridin-2-yl)-4-oxobutanamide
3-(1-butyl-1H-imidazol-2-yl)-N-(3-cyanophenyl)piperidine-1-carboxamide
4-{5-[3-(difluoromethoxy)phenyl]-3-methyl-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
N-({1-[(3-ethenylphenyl)methyl]pyrrolidin-3-yl}methyl)pyrrolidine-1-sulfonamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(pyrrolidin-3-yl)benzamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
4-methoxy-N-(oxan-4-yl)-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
2-(dimethylamino)-N-methyl-N-(2-phenoxyethyl)-2,3-dihydro-1H-indene-2-carboxamide
6-methyl-3-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-1,2-dihydroquinolin-2-one
N-(dimethyl-1,2-oxazol-4-yl)-5-[1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[1-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(3-hydroxy-2,2-dimethylpropyl)piperidine-4-carboxamide
N-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
3-[(4aR,7aS)-4-(4-chlorobenzoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-pyrrole-3-carboxamide
3-{1-[(2S)-oxolane-2-carbonyl]azetidin-3-yl}pyridine
2-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]pyridine-4-carboxylic acid
N-[2-(diethylamino)ethyl]-4-methoxy-N-methyl-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
5-tert-butyl-4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}furan-2-carboxamide
4-(6-methoxypyridin-2-yl)-2-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenol
5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine
5-[benzyl(methyl)amino]-2-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,3-dihydropyridazin-3-one
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-{1-methyl-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
2-(2-{[(4-fluorophenyl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-methyl-4-({5-[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}acetamide
2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)isoquinoline
methyl 4-[({3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}carbamoyl)amino]benzoate
(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-1-cyclopropanecarbonyl-decahydro-1,6-naphthyridine
2-[(1-acetylpiperidin-3-yl)amino]-N,N-bis(prop-2-en-1-yl)acetamide
2-[(4-methoxyphenyl)methyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-amino-3-ethyl-N-[1-(oxan-4-yl)piperidin-4-yl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(2,3-dimethoxyphenyl)-1-[3-(1H-imidazol-5-yl)phenyl]-1H-imidazole
7-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
methyl 2-({7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazol-5-yl}formamido)-4-(methylsulfanyl)butanoate