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N-ethyl-5-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]pyrimidin-2-amine
ethyl 4-[(2-chlorophenyl)methyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxylate
4-(2-amino-6-methylpyrimidin-4-yl)-N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)piperazine-1-carboxamide
2-[6-(4-fluorophenyl)pyridazin-3-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-4-methyl-1H-imidazole-5-carboxamide
(1-methyl-5-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-ethoxypropanamide
2-{4-[5-(4-methoxyphenyl)furan-2-carbonyl]morpholin-3-yl}acetic acid
4-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridin-2-amine
1-[6-(4-methylpiperidin-1-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-{2-[cyclopentyl(methyl)amino]ethyl}-N-methyl-2-oxo-1-phenylpyrrolidine-3-carboxamide
8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-amino-N-(5-chloro-2-ethyl-3-methyl-1-benzofuran-7-yl)pyrrolidine-1-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1-ethyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(4-ethylphenoxy)ethyl]-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-{2-[2-(dimethylamino)-2-(2-fluorophenyl)acetamido]ethyl}-2-methylpropanamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-[(4-hydroxy-3-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
3-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-N-methylbenzamide
7-(cyclopropylmethyl)-6-(2,5-dimethylfuran-3-yl)-N-ethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-cyclopentyl-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-(1,3-benzothiazol-2-yl)-N-(thian-4-yl)piperidin-3-amine
N-(cyclohexylmethyl)-2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidin-3-yl]methanol
1-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-3-(1,1-dioxo-1λ6-thiolan-3-yl)urea
N4-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-6-(propan-2-yl)pyrimidine-2,4-diamine
2-(4-amino-1H-pyrazol-1-yl)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]acetamide
1-(pyridin-4-ylmethyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
N-[4-(2-methoxyphenyl)phenyl]-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
(7S,9aR)-7-benzyl-6,9-dioxo-N-phenyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-(3,5-dimethoxyphenyl)-3-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}propanamide
1-(2-methoxyethyl)-N-[2-(5-methylfuran-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
5-(1-cyclohexyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)-N-(propan-2-yl)pyrimidin-2-amine
{1-[(2-methyl-1,3-thiazol-5-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
2-[({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)methyl]-3,4-dihydroquinazolin-4-one
3-{[(furan-2-ylmethyl)(methyl)amino]methyl}-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-(3,4-dimethoxyphenyl)-N,N-dimethylbenzamide
2-(4-{[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}-6-methylpyrimidin-2-yl)phenol
5-chloro-2-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]phenol
3-(2-fluorophenyl)-4-{1H-imidazo[4,5-c]pyridin-2-yl}-1-methyl-1H-pyrazole
N-[2-(4-chlorophenyl)propyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
{imidazo[1,2-a]pyridin-3-ylmethyl}(methyl){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
1-(4-methylpiperidin-1-yl)-2-{2-[1-(pyridin-3-yl)-1H-imidazol-2-yl]phenoxy}ethan-1-one
2-(1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}azetidin-3-yl)pyridine
1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]-5-oxopyrrolidine-3-carboxylic acid
2-(4-chloro-1H-pyrazol-1-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
(2R,6S)-4-{6-chloro-3-[(4-methoxypiperidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}-2,6-dimethylmorpholine
8-methoxy-N-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine