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1-butyl-4-(2-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-2-oxo-1-phenylethyl)piperazine-2,3-dione
2-{4-[(4-acetylpiperazin-1-yl)methyl]-1,2,3,6-tetrahydropyridin-1-yl}-N-cyclopropylacetamide
4-(hydroxymethyl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]pyridine-2-carboxamide
(3R,4R)-4-{[6-(morpholine-4-carbonyl)pyrazin-2-yl]amino}piperidin-3-ol
3-[(2R,3R,6R)-5-[(2E)-3-phenylprop-2-en-1-yl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})(pyrimidin-4-ylmethyl)amine
6-(4-carbamoylpiperidin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-ethyl-5-{1-[5-(5-methylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl]amino)ethan-1-ol
N4-(2-ethoxybutyl)-6-(propan-2-yl)pyrimidine-2,4-diamine
3-({1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
4-[4-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)phenyl]but-3-yn-1-ol
2-[({2-[4-(morpholin-4-yl)butoxy]phenyl}methyl)amino]acetamide
ethyl 4-({[3-(1H-pyrazol-5-yl)phenyl]carbamoyl}amino)piperidine-1-carboxylate
(2S)-2-({5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazol-3-yl}formamido)propanamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-phenoxybenzamide
3-[(2-aminopyrimidin-5-yl)methyl]-3-methyl-1-[2-(morpholin-4-ylmethyl)phenyl]urea
2-(cyclopropylmethyl)-9-(2-methyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
3-(1H-1,3-benzodiazol-1-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]ethan-1-one
2-{imidazo[1,2-a]pyridin-3-yl}-1-[4-(2-methoxyphenoxy)piperidin-1-yl]ethan-1-one
{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(1H-pyrazol-5-ylmethyl)-1,2-oxazole-3-carboxamide
N-(1,2,3-thiadiazol-5-yl)-3-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}benzamide
(4aS,8aR)-1-butyl-2-oxo-N-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridine-6-carboxamide
methyl 2-[(3S,4R)-3-methanesulfonamido-4-propylpyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxylate
N-{[7-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
4-[2-(2-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}phenoxy)ethyl]morpholine
7-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-{1-[(3-chlorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}-1-methyl-1,2-dihydropyridin-2-one
1-[1-(2,2-difluoroethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-(3-fluoropyridin-4-yl)-3-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)benzamide
2-[(5-hydroxypyrazin-2-yl)formamido]-N-(2-methoxy-5-methylphenyl)acetamide
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
(3S,4R)-4-(3-fluorophenyl)-1-[4-(morpholin-4-yl)butanoyl]pyrrolidine-3-carboxylic acid
5-(2-chloro-4-fluorophenoxymethyl)-3-(3-cyclohexylpyrrolidine-1-carbonyl)-1,2-oxazole
3-{1-[2-(1H-indol-3-yl)acetyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
3-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]sulfamoyl}-N-(oxolan-3-ylmethyl)benzamide
3-methyl-N-[2-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propyl]thiophene-2-carboxamide
1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidin-3-amine
4-methyl-6-{4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}pyrimidin-2-amine
4-methyl-2-[1-(pyridazine-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-methyl-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
2-amino-6-tert-butyl-4-[2-(2-hydroxyethoxy)phenyl]pyridine-3-carbonitrile
N-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-5-propyl-1,3,4-oxadiazol-2-amine
1-(2-methylpropyl)-4-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-1,4-diazepane
1-(2-{4-[(2Z)-3-(3-fluorophenyl)prop-2-enoyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(3-methylphenyl)-1H-indazol-1-yl]acetamide
(3aR,6aR)-2-(2-methylbenzoyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid