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1-(2-chloro-4,6-dimethylphenyl)-3-(1-methyl-2-oxopyrrolidin-3-yl)urea
3-{4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-1H-pyrazol-1-yl}propanoic acid
(2S,4R)-4-amino-N-ethyl-1-[4-(1H-imidazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
1-(4-fluorophenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]cyclopropane-1-carboxamide
ethyl 1-(3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)piperidine-3-carboxylate
N-cyclopentyl-3-[5-(4-methylpentanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(propan-2-yl)piperidine
1-{3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-[2-(methylsulfanyl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
(5-{1-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
4-(1-methyl-1H-indole-4-carbonyl)-1,4-oxazepan-6-ol
(1R,9aR)-1-[({[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
ethyl 4-[1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]piperazine-1-carboxylate
5-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
2-{[propyl(pyridin-4-ylmethyl)amino]methyl}pyridine-3-carboxylic acid
3-(2-chlorophenyl)-1-methyl-3-{2-oxo-2-[3-(pyridine-3-carbonyl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
3-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-2,3-dihydro-1H-inden-1-one
5-[(4-ethoxypiperidin-1-yl)methyl]-2-methoxybenzoic acid
8-(3-methylbutanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
5-(3,4-dimethoxyphenyl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1,2,4-triazin-3-amine
2-(2-methylpropyl)-6-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(1R,5R)-6-(cyclopropylmethyl)-3-(1,5-dimethyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
(1S,5R)-3-(6-aminopyridine-3-carbonyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3S,5S)-1-ethyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
(1S,5R)-3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,3S)-7-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
2-(5-chloro-2-methoxyphenyl)-N,N,5-trimethylpyrimidin-4-amine
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
1-(2-ethoxyphenyl)-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazine
[4-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-1,4-oxazepan-6-yl]methanol
(2E)-N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(4-methoxyphenyl)prop-2-enamide
5-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-methyl-N-{2-[(4-phenylbutan-2-yl)amino]ethyl}methanesulfonamide
N-(diphenylmethyl)-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
7,7-dimethyl-2-[4-(methylsulfanyl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2-(furan-2-ylmethyl)propan-1-ol
N-butyl-3-({[3-(trifluoromethyl)phenyl]formamido}methyl)piperidine-1-carboxamide
9-[2-hydroxy-4-(methylsulfanyl)butanoyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[1-(piperidin-1-yl)ethyl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)furan-2-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]oxolane-3-carboxamide
2-[(3-fluorophenyl)methyl]-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]morpholine
7-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyrimidin-4-yl}pyrrolidin-3-ol
N-[2-(4-chlorophenyl)ethyl]-3-(2-methoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-(2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetyl)-1,4-diazepan-5-one
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-methoxyethan-1-one
7-fluoro-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-[2-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one