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5-chloro-N-ethyl-N-(oxan-4-ylmethyl)pyridine-2-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-2-(1-ethyl-1H-pyrazol-4-yl)quinoline
[4-({1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
(1S,2S,9R)-11-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
5-chloro-N-(1-propylcyclopropyl)pyridine-3-carboxamide
N-(4-{4-[4-(2-methoxyethyl)piperazin-1-yl]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]propanamide
4-(4-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidine-1-carbonyl}phenyl)-2-methylbut-3-yn-2-ol
2-{2-[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-cyclohexyl-N-[cyclopropyl(6-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
3-(methylsulfanyl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)propanamide
2-[(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-6-methylpyridine
N-(2,3-dimethylphenyl)-N'-(3-phenylprop-2-yn-1-yl)-N'-(prop-2-en-1-yl)propanediamide
4-(1H-imidazol-1-ylmethyl)-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-ol
1-benzyl-6-[(2-hydroxy-6-methoxyphenyl)methyl]-3-(2-methoxyphenyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-(piperidin-1-ylmethyl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-ol
(4aS,8aR)-6-(4-methoxy-2-methylbenzoyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}urea
2-(4-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}morpholin-2-yl)ethan-1-ol
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(3S,9aR)-8-benzyl-3-[(1R)-1-(benzyloxy)ethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,7aR)-1-(1-aminocyclopropanecarbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-methyl-N2-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidine-2,4-diamine
[(1,5-dimethyl-1H-indazol-3-yl)methyl](5-methylhex-5-en-2-yl)amine
(1S,5R)-3-[(2-aminopyridin-3-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-benzyl-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,3-benzoxazole-5-carboxamide
1-(4-fluorophenyl)-N-[3-(1H-indazol-1-yl)propyl]cyclopropane-1-carboxamide
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{1-[4-(pyridin-3-yloxy)phenyl]-1H-imidazol-2-yl}pyridine
6-(benzylamino)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-9-(5-methylpyrazine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-{[(1H-imidazol-2-ylmethyl)amino]methyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
4-(1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)quinoline
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)-5-methoxy-1,4-dihydropyridin-4-one
[2-(isoquinolin-1-yloxy)hex-5-en-1-yl](methyl)(pyridin-3-ylmethyl)amine
1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
5-propyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-3-(piperazin-1-yl)propan-1-one
N,1-dimethyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-N-methylpyrrolidine-2-carboxamide
3-{[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{3-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-methyl-1H-indole-6-carboxamide
1-methanesulfonyl-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
N-(2-methoxyethyl)-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}piperidine-3-carboxamide
N-(2,4-difluorophenyl)-9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)oxane-4-carboxamide
N-{1-[4-(2-methylphenyl)phenyl]ethyl}acetamide