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3-[(2-fluoroethyl)sulfamoyl]-N-[2-(1,3-thiazol-2-yl)ethyl]benzamide
N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(pyridin-4-ylsulfanyl)acetamide
(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-[(2-methylphenyl)methyl]piperidin-3-yl)methanol
2,5-dimethyl-4-(4-{[4-(pyridin-2-yl)phenyl]methyl}piperazin-1-yl)pyrimidine
2-[4-(4-ethyl-5-methylthiophene-3-carbonyl)-1-methylpiperazin-2-yl]ethan-1-ol
4-chloro-1-methyl-3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1H-indazole
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
4-(3-fluorophenoxy)-1-[(2R)-oxolane-2-carbonyl]piperidine
1-[1-(4-fluorobenzoyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
1-[(6-hydroxynaphthalen-2-yl)methyl]piperidine-3-carbonitrile
1-(2-methyl-4-{[2-(morpholin-4-yl)butyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N2,N2,5,6-tetramethyl-N4-{pyrazolo[1,5-a]pyridin-3-ylmethyl}pyrimidine-2,4-diamine
4-[2-(pyridin-2-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
2-(1H-pyrazol-1-yl)-1-[4-(pyridin-3-yl)piperazin-1-yl]butan-1-one
N-[3-({[1-(4-methoxyphenyl)propan-2-yl]amino}methyl)-5-(pyrrolidine-1-carbonyl)phenyl]acetamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
8-(2,6-dimethylpyridin-4-yl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyridine-3-carboxamide
1-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-[(4,6-dimethylquinolin-2-yl)sulfanyl]-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
2-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(3S,4R)-4-(3-methoxyphenyl)-1-(1-phenylcyclopropanecarbonyl)pyrrolidine-3-carboxylic acid
propyl 1-methyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-carboxylate
4-({1-[3-(4-hydroxyphenyl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
(3aS,7aR)-2-(3-fluoropyridine-2-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
7-[4-(trifluoromethyl)benzenesulfonyl]-2-oxa-7-azaspiro[4.5]decane
N-[4-(4-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]-2-fluorobenzamide
ethyl 4-[6-(1-benzofuran-2-carbonyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
4,6-dimethyl-2-({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)pyridine-3-carbonitrile
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[2-(7-methyl-1H-indol-3-yl)ethyl]propanamide
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
1-[1-ethyl-5-(1,2,5-thiadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
3-[(3R,4S)-1-(2-ethoxybenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(6-methylpyridine-3-carbonyl)pyrrolidin-3-yl]methanol
N-[(2S,4R,6S)-2-benzyl-6-(4-ethoxyphenyl)oxan-4-yl]acetamide
(2R,3R)-3-[(2-hydroxyethyl)(methyl)amino]-1'-[(3-methyl-1H-pyrazol-5-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
4-(4-methoxynaphthalen-1-yl)-3-methyl-4H,5H,6H,7H-[1,2]oxazolo[5,4-b]pyridin-6-one
1-(cyclopentylcarbamoyl)-4-phenoxypiperidine-4-carboxylic acid
1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
methyl (2R,4S)-4-hydroxy-1-(quinoxaline-2-carbonyl)piperidine-2-carboxylate
2-{[3-(diethylamino)pyrrolidin-1-yl]methyl}-6-fluoroquinolin-4-ol
N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-4-(1H-1,2,4-triazol-3-yl)benzamide
2-{1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-3-yl}-1,3-benzothiazole
3-(1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)propanamide
N3-butyl-N5-[(4-fluorophenyl)methyl]-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-{ethyl[2-(4-methylbenzenesulfonyl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
2-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)benzonitrile
3-phenyl-1-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)propan-1-ol