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3-{2-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
1,7-dimethyl-2-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-indole
(2E)-1-{4-[(3-hydroxypropyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-phenylprop-2-en-1-one
(1R,3S)-7-[2-(3,4-dimethylphenoxy)ethyl]-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-ethylpiperazin-1-yl)acetamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(dimethylamino)-2-(3-methylphenyl)acetamide
9-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-methyl-N-[2-phenyl-2-(piperidin-1-yl)ethyl]pyrimidin-2-amine
4-{1-[1-(3-methoxyphenyl)piperidin-4-yl]azetidin-3-yl}pyridine
2-[(oxan-3-yl)amino]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-{[(1H-imidazol-2-ylmethyl)(methyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(oxan-2-ylmethoxy)ethan-1-one
methyl 3-[propyl(pyridin-3-ylmethyl)carbamoyl]propanoate
7-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-2-(3-methoxypiperidin-1-yl)pyridine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidin-2-amine
2-[(4-benzylpiperazin-1-yl)methyl]-N-(1,4-dioxan-2-ylmethyl)-1,3-oxazole-4-carboxamide
9-(2-methoxyethyl)-4-[(3-methoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
1-(4-{[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
2-(6-methoxynaphthalen-2-yl)-4-(4-methylpiperidine-4-carbonyl)morpholine
N-(1H-indol-6-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-2-(methylamino)-N-{3-[(4-methylphenyl)sulfanyl]propyl}pyrimidine-5-carboxamide
N-[4-(pyridin-2-ylmethoxy)phenyl]-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
2-(1-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]-5,6,7,8-tetrahydroquinazolin-2-amine
2-{[5-(2-amino-3-cyano-6-phenylpyridin-4-yl)pyrimidin-2-yl]amino}acetic acid
1-(3-methylpyridin-4-yl)-4-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1,4-diazepane
7-methoxy-3-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-2,3,4,5-tetrahydro-1H-3-benzazepine
3-(5-methylfuran-2-yl)-N-(2-oxoazepan-3-yl)-1H-pyrazole-5-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}but-2-ynamide
(1S,5R)-3-(4-cyclobutyl-6-methylpyrimidin-2-yl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2H-1,2,3-benzotriazol-2-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}acetamide
5-methanesulfonyl-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
N-butyl-N-[(5-methylthiophen-2-yl)methyl]-1-propyl-1H-pyrazole-5-carboxamide
N3-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-benzyl-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1R,7S)-3-cycloheptyl-6-[3-(piperidin-1-yl)azetidine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-[2-(4-ethylphenoxy)ethyl]-N-methyl-2-(3-methyl-1,2-oxazol-5-yl)acetamide
2-{4-[4-(3,4-difluorobenzoyl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
N-(pyrrolidin-3-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
(3aS,6aS)-2-[(2-chlorophenyl)methanesulfonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-3-ene-1-carboxamide
3-(3-fluorophenyl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
3-(1,3-dimethyl-1H-pyrazol-5-yl)-4-(furan-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(3,6-dimethylpyrazin-2-yl)-4-(1H-imidazol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(2-amino-5,6-dimethylpyrimidin-4-yl)amino]-N-phenylpropanamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(methylsulfanyl)acetamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane