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5-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-5-(pyridin-3-yl)imidazolidine-2,4-dione
1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-ethyl-N-[(3-phenylphenyl)methyl]piperidine-4-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(2-oxopiperidin-1-yl)ethyl]benzamide
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyridin-2-amine
methyl 3-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)carbamoyl)propanoate
1-benzyl-N-methyl-5-(prop-2-en-1-yl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N,N,8-trimethyl-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
4-[2-(1H-pyrazol-1-yl)ethyl]-1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidine
3-{2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
5-(2-phenylethyl)-4-propyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-(2-{1-[2-(difluoromethoxy)benzoyl]piperidin-2-yl}ethyl)morpholine
2-(isoquinolin-5-yl)-3-methoxypyridin-4-amine
2-[2-methyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]acetic acid
8-methoxy-N-[2-(N-methylmethanesulfonamido)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-methanesulfonyl-2-methyl-N-[1-(thiophen-3-yl)propan-2-yl]pyrimidin-4-amine
N-phenyl-1-(1-phenylcyclopropanecarbonyl)piperidin-3-amine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
8-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{2-[(3-chloro-4-fluorophenyl)carbamoyl]acetyl}piperidine-3-carboxylic acid
(4aR,7aS)-1-acetyl-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1H-imidazol-2-ylmethyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-methoxy-2-phenyl-1-(7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-phenyl-1-{1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-4-yl}ethan-1-ol
N-[(2S)-pyrrolidin-2-ylmethyl]-3-[(2,2,2-trifluoroethyl)sulfamoyl]benzamide
(1R,7S)-N-(1H-imidazol-2-ylmethyl)-N-methyl-4-oxo-3-(2-phenoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)pyridine-2-carboxamide
1-[3-(3-chlorophenoxy)azetidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
2-methoxy-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]acetamide
4-benzyl-3-[1-(5-hydroxypyrazine-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2,5-dihydro-1H-pyrrole-1-carbonyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine
3-(2-amino-1,3-thiazol-4-yl)-N-[(2,4,5-trifluorophenyl)methyl]propanamide
4-[(1-benzothiophen-2-ylmethyl)amino]-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-(2-ethylpyrrolidin-1-yl)-3-(2-methyl-1H-indol-1-yl)propan-1-one
1-[4-({4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}methyl)phenyl]ethan-1-one
5-{[3-(2-oxopyrrolidin-1-yl)propyl]carbamoyl}-1H-imidazole-4-carboxylic acid
1-{[4-(2-methylpropyl)phenyl]methyl}-N-(1,3-thiazol-2-ylmethyl)piperidin-3-amine
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-2-[3-(methoxymethyl)pyrrolidin-1-yl]pyrimidine
(3R,7S,8aS)-7-{[(3,4-difluorophenyl)methyl]amino}-3-[(1S)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4,6-dimethylpyridine-3-carbonitrile
5-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]quinoxaline
6-{[(2,2-dimethyloxan-4-yl)(ethyl)amino]methyl}pyridine-2-carboxylic acid
N-(1-cyclopropylethyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
4-(2,5-dimethoxyphenyl)-2-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenol
1-[2-(dimethylamino)ethyl]-6-oxo-N-[(1-phenylcyclopentyl)methyl]piperidine-3-carboxamide
N-benzyl-N,1-dimethyl-5-{[3-(propan-2-yloxy)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-cyclopropyl-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-6-oxopiperidine-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[3-(methylsulfanyl)propyl]piperidin-3-yl}piperazine