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2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
2-(dimethyl-1,3-thiazol-4-yl)-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
2-[5-(2-methyl-3-phenylcycloprop-2-en-1-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
3-methyl-5-{2-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(2-{[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]methyl}-4-(pyrazin-2-yl)phenoxy)acetic acid
7-(2,2-dimethylpropyl)-2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
5-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1H-indole
4-[(2,6-dichlorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
5-methyl-2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N-(4-{[ethyl(oxolan-2-ylmethyl)amino]methyl}phenyl)acetamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
N-{3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}acetamide
4-{2-oxo-2-[3-(pyridin-2-yloxy)piperidin-1-yl]ethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
5-{1H-pyrazolo[3,4-b]pyridin-1-yl}-N-(pyridin-3-yl)furan-2-carboxamide
1-(2-fluorophenyl)-3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}urea
5-(hydroxymethyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]furan-2-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-ol
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-4-phenylbutane-1,4-dione
2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-ylmethyl]-3,5-dimethyl-1,4-dihydropyridin-4-one
N-methyl-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
(2E)-N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-3-(3-fluorophenyl)-N-(oxolan-2-ylmethyl)prop-2-enamide
4-(7-methyl-1H-indol-3-yl)-2-(1,2-oxazol-5-yl)phenol
1-(4-methoxyphenyl)-4-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}butane-1,4-dione
6-cyclopentyl-N,1-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
2-[methyl({5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl})amino]-1-phenylethan-1-ol
1-(2-ethoxyphenyl)-3-[2-(ethylsulfanyl)ethyl]urea
8-methyl-3-{2-[methyl(2-methylpropyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-cyclopropylpyrimidine-5-carboxamide
1-(1-propyl-1H-pyrazole-5-carbonyl)-2-(pyrrolidine-1-carbonyl)piperazine
2-methoxy-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}pyridine-4-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(3-methylthiophen-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-methyl-1,3-thiazole-5-carbonyl)-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-oxo-1,2-dihydroquinolin-1-yl)acetamide
(3S,5R)-5-(morpholine-4-carbonyl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
4-{[(3-chloro-4,5-dimethoxyphenyl)methyl]amino}-1-(2,2-dimethylpropyl)pyrrolidin-2-one
{4-[(3-fluorophenyl)methyl]-1-(oxolane-3-carbonyl)piperidin-4-yl}methanol
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(5-methylthiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-benzyl-N-(1,3-thiazol-2-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
1-(3-{5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-2-phenoxyethan-1-one
N-[(2,5-dimethoxyphenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
N-(1-hydroxybutan-2-yl)-2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)-N-(thiophen-3-ylmethyl)acetamide
5-chloro-N-[(4-fluorophenyl)methyl]-6-oxo-N-(oxolan-2-ylmethyl)-1,6-dihydropyridine-3-carboxamide
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one