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3-[1-(3-cyanopyridin-2-yl)piperidin-3-yl]-N-[(3,4-difluorophenyl)methyl]propanamide
N-cyclopropyl-3-(3-methyl-1H-pyrazol-1-yl)-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}propanamide
N-(2,4-dimethoxyphenyl)-3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}propanamide
N2-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrimidine-2,4-diamine
7-[2-(propan-2-yloxy)phenyl]pyrazolo[1,5-a]pyridine
5-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-propyl-1,2,4-oxadiazole
4-(4-fluorophenyl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-1,2,3,6-tetrahydropyridine
2-(3-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)-1,3-thiazole
methyl 3-[(3S,4R)-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]propanoate
N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-(3-propyl-1H-pyrazole-4-carbonyl)piperazin-2-one
2-(2-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)pyridine
methyl({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})[2-(oxan-2-yl)ethyl]amine
2-{1-[(3,4-difluorophenyl)methyl]-4-(1H-indol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-3-methyl-1,2-dihydroquinoxalin-2-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
1-{2-[(4-fluoropiperidin-1-yl)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
2-{[4-(naphthalen-1-yl)-5-(pyridin-3-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-cyclopentyl-1-methyl-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1R,5R)-6-benzyl-3-(2,6-dimethoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[5-(4-methyl-1H-imidazol-5-yl)-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
5-fluoro-2-[1-(1,2-oxazole-3-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
(5-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
N-(3,3-diphenylpropyl)-2-(morpholin-3-yl)acetamide
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
(1R,5R)-6-[(3,4-difluorophenyl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-methyl-5-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,3-thiadiazole
2-[3-methyl-4-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrazol-1-yl]ethan-1-ol
methyl 8-[3-(methylsulfanyl)propyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(2,2-dimethyloxan-4-yl)-N-ethyl-2-(4-methyl-1,4-diazepan-1-yl)acetamide
[4-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)morpholin-3-yl]methanol
2-methoxy-1-{4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,7S)-6-(3-oxopiperazine-1-carbonyl)-3-(2-phenoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1,3-dimethyl-5-({[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(5-methylthiophen-2-yl)methyl]amine
5-[(4-fluorophenyl)methyl]-3-(3-hydroxypropyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
(2-methoxyethyl)(oxolan-2-ylmethyl)[(5-phenylthiophen-2-yl)methyl]amine
7-chloro-2-methyl-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(4-hydroxyphenyl)-N-methyl-2-phenylpropanamide
2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-(hydroxymethyl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-3-ol
3-{1-[5-(ethylsulfanyl)thiophene-2-carbonyl]piperidin-3-yl}benzoic acid
3-(2H-1,3-benzodioxole-5-carbonyl)-1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidine
3-(2-methoxyphenyl)-3-{2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
3-{[2-(N-methylmethanesulfonamido)ethyl]sulfamoyl}-N-(prop-2-en-1-yl)benzamide
2-(1-{[1-(propane-2-sulfonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-butyl-3-methoxy-N-[(3-methylthiophen-2-yl)methyl]propanamide
4-(2-ethoxyphenyl)-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}piperazine-1-carboxamide