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3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]propan-1-ol
5-{3-[1-(dimethylamino)ethyl]phenyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(4-{[(1R,2S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecan-11-yl]methyl}phenoxy)acetic acid
N-[(2-chlorophenyl)methyl]-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]propanamide
(4aS,7aR)-1-(2-methoxy-6-methylbenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(carbamoylamino)-N-[1-(cyclohexylmethyl)piperidin-3-yl]acetamide
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-[(4aR,7aS)-4-[(2-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-amino-N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
8-methoxy-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(2-methoxyacetamido)-5-[(pentan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[1-(5-methoxy-1H-indole-2-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
(3R,4S)-4-cyclopropyl-1-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}pyrrolidin-3-amine
1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-(4-methyl-1-phenylpentyl)urea
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]urea
2-[2-(dimethylamino)ethyl]-9-(3-propyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-acetamido-N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-3-(1H-imidazol-4-yl)propanamide
3-(furan-2-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
N-(1-methyl-1H-indazol-6-yl)azocane-1-carboxamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-(butan-2-yl)-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]cyclopentanamine
1-({1-[(4-acetamidophenyl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
2,6,8-trimethyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}quinoline-4-carboxamide
2-[2-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)phenoxy]acetamide
(isoquinolin-5-ylmethyl)(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
3-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]-1,3-oxazolidin-2-one
3-(4-hydroxyphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]propan-1-one
N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-3-(4-methylphenyl)propanamide
N-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-methyl-N-{[6-methyl-2-(2-methylphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
N-benzyl-N-methyl-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-amine
2-(8-methoxyquinolin-5-yl)-5,6-dimethylpyridine-3-carbonitrile
methyl 3-[(3S,4R)-1-[(4-methoxy-3-methylphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
6-methoxy-3-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydroquinazolin-4-one
4-cyano-N-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
N-(3-chloro-4-propanamidophenyl)-3-methyl-1H-pyrazole-5-carboxamide
2-amino-N-[1-(4-methoxyphenyl)-4-(pyridin-3-yloxy)-1H-indazol-3-yl]acetamide
ethyl 4-(1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
2-(2-{[4-(difluoromethoxy)phenyl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)-6-methylpyridine
5-acetyl-N-[(2-benzyl-1,3-thiazol-4-yl)methyl]thiophene-2-carboxamide
1-cyclohexyl-4-[(4-fluorophenyl)methyl]-1,4-diazepan-5-one
2-({[2-(dimethylamino)ethyl][(3-methylthiophen-2-yl)methyl]amino}methyl)-6-methylpyridin-3-ol
5-[(4-benzylpiperidin-1-yl)methyl]-N-(1,2-oxazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]acetamide
3-methyl-7-[4-(4-methylphenoxy)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
methyl 2-{N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamido}acetate
N-cyclopropyl-1-[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane