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2-methyl-4-(3-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}phenyl)butan-2-ol
1-(3-methylpiperidin-1-yl)-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-methanesulfonamido-N-[(3R,4S)-1-[(5-methylfuran-2-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
1-cyclohexanecarbonyl-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrrolidine-2-carboxamide
3-{[1-(2,5-dihydro-1H-pyrrole-2-carbonyl)piperidin-4-yl]methyl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[7-(piperidin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine
(3R,4S)-1-(3-chloro-4-propoxybenzoyl)-4-cyclopropylpyrrolidin-3-amine
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2,2-diphenylacetamide
2-(2,4-difluorophenyl)-5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)pyrrolidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
3-(1H-indol-5-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
5-cyclopropyl-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1,3,4-oxadiazol-2-amine
methyl (2S,4R)-1-(1-benzylpiperidin-4-yl)-4-{2-[3-(trifluoromethyl)phenyl]acetamido}pyrrolidine-2-carboxylate
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
1-(5-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
1-{[1-(6-{[2-(dimethylamino)ethyl](methyl)amino}pyridine-3-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,2-diphenylacetamide
2-methoxy-4-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyridine
(3aR,6aS)-2-[4-(5-methylfuran-2-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole
N-(1-cyclopentanecarbonylpiperidin-4-yl)-4-(piperidin-3-yl)benzamide
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
4-(1H-imidazol-1-yl)-N-(2-methylpropyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
2-{[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]methyl}-4-oxo-1,4-dihydroquinoline-6-carboxamide
N3-[2-(2,4-dichlorophenyl)ethyl]piperidine-1,3-dicarboxamide
8-(1-hydroxypropan-2-yl)-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}azepan-2-one
3-(2-{[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}propyl)-3,4-dihydroquinazolin-4-one
2-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-4,6-dimethylpyridine-3-carbonitrile
1-ethyl-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-1H-pyrazole-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-(9H-purin-6-yl)piperazin-2-one
2-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidine-3-carbonyl)pyridine
2-(1H-pyrazol-1-ylmethyl)-4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-1,4-oxazepane
9-[2-(1,2-benzoxazol-3-yl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
4-(cyclohexylmethyl)-11-{[2-(2-fluorophenyl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(2R)-2-amino-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-phenylacetamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-[(2-methoxyphenyl)methyl]pyrimidine
N-[(5-ethylpyridin-2-yl)methyl]-2-hydroxy-N-methyl-3-(2-methylphenoxy)propanamide
3-[4-(4-methylpyrimidin-2-yl)piperazin-1-yl]-1,2-benzothiazole
2-(5-{[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]methyl}furan-2-yl)benzonitrile
2-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-8-methyl-2,8-diazaspiro[5.5]undecane
N-{2-[(2,3,6-trimethylquinolin-4-yl)formamido]ethyl}pyridine-3-carboxamide
4-({5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}amino)-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
N-[4-(4-{[2-(1H-indol-3-yl)ethyl]amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
(1R,3S)-3-amino-N-[(3-methoxyphenyl)methyl]-N-(3-methoxypropyl)cyclohexane-1-carboxamide
1-{3-[4-(3-methylphenoxy)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methyl-5-{2-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-chloro-4-fluorobenzamide
5-amino-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1H-pyrazole-3-carboxamide
(2S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide