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3-methyl-7-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(pyridin-2-yl)piperazine
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-(oxolan-2-ylmethoxy)acetamide
2-[4-benzyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-methyl-N-(propan-2-yl)acetamide
1-cyclopropanecarbonyl-N-[3-(1H-indazol-1-yl)propyl]piperidine-4-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-3-[2-oxo-2-(piperidin-1-yl)ethoxy]benzamide
(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-{[(3-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-(4-fluorophenyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]benzamide
(2R,6R)-10-methoxy-4-(3-propyl-1H-pyrazole-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[2-(2-fluorophenyl)-1-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl}ethyl]-N-methylthiophene-3-carboxamide
(3S)-N-tert-butyl-2-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(cyclohexylsulfamoyl)-5-(pyrimidin-5-yl)benzoic acid
3-chloro-N-[(3S,4S)-1-ethyl-4-methoxypyrrolidin-3-yl]-4-fluoro-1-benzothiophene-2-carboxamide
3-ethyl-1-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]urea
4-(3,5-difluoropyridine-2-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]amine
(1R,5S,8S)-8-methoxy-N-[4-methoxy-3-(2-methoxyacetamido)phenyl]-3-azabicyclo[3.2.1]octane-3-carboxamide
6-methyl-2-(4-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(3S,4R)-1-[2-(difluoromethoxy)benzoyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
N-(2-methoxyethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[3-(4-{[cyclopropyl(ethyl)amino]methyl}-2-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
3-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-[3-(prop-2-en-1-yloxy)phenyl]urea
6-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine-2-carboxamide
(4-{4-[1-(1H-indol-4-ylmethyl)pyrrolidin-3-yl]pyridin-2-yl}phenyl)methanol
methyl 3-chloro-4-{[3-(propoxymethyl)pyrrolidine-1-carbonyl]amino}benzoate
1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N,5-dimethyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[1-(methoxymethyl)cyclopropyl]methyl}acetamide
1-{3-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
3-[2-(4-fluorophenyl)ethyl]-1-(1,2-oxazole-3-carbonyl)piperidine
methyl 3-{[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}propanoate
3-(2-butylpyrrolidine-1-carbonyl)-5-(2,4-difluorophenoxymethyl)-1,2-oxazole
2-(1-methyl-1H-pyrazol-3-yl)-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
2-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methoxybenzamide
4-{[5-(3,4-dimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
3-[(3-carbamoylphenyl)methyl]-N-cyclohexylpyrrolidine-1-carboxamide
methyl(pyridin-3-ylmethyl){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
2-[(3,4-dimethoxyphenyl)methyl]-6-(piperidine-1-carbonyl)-1,3-benzoxazole
(3R,4S)-4-(5-methylfuran-2-yl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)pyrrolidin-3-amine
1-{2-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
5-(5-methyl-1,3-oxazol-4-yl)-1-(propan-2-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
5-(4-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
1-({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)cyclopentane-1-carboxamide
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3-benzothiazole-5-carboxamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(cyclopropylmethyl)piperazine
3-(2-methoxyethyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
N-(cyclohex-1-en-1-ylmethyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-3-(4H-1,2,4-triazol-3-yl)piperidine
methyl 4-(2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)butanoate
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(4,6-dimethylpyridine-3-carbonyl)pyrrolidin-3-yl]methanol