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2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-6,7-dimethoxyquinazolin-4-amine
1-(2-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
1-ethyl-3,5-dimethyl-4-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1H-pyrazole
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[2-(propan-2-yl)pyrimidine-4-carbonyl]-decahydro-1,6-naphthyridin-2-one
N,1,3-trimethyl-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-(4-phenylbutan-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(1H-indazol-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
(1H-1,3-benzodiazol-2-ylmethyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine
7-(3-chloropyridine-4-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-benzyl[(1H-indazol-6-yl)amino]sulfonamide
2-methyl-6-(1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
5-ethyl-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
methyl 8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(4aS,7aR)-1-pentanoyl-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[3-(2-methylpyridine-3-carbonyl)-9-(pyridin-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-(2-hydroxyethyl)-N-methyl-2-phenylacetamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-ethyl-3-methylpiperidine-3-carboxamide
1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
N-methyl-5-(propan-2-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-({3-[(3-chlorophenyl)methyl]-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl}methyl)acetamide
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl})(thiophen-3-ylmethyl)amine
3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-[4-(morpholin-4-ylmethyl)phenyl]urea
6-cyclopentyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carboxamide
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-[(4-methylphenyl)amino]-2-phenylpropanamide
1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
(3S,4R)-1-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
methyl 1-[(3R,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
(4aS,7aR)-1-(1-aminocyclopropanecarbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-ethyl-5-[4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1,2,4-oxadiazole
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amine
3-(5-{[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-1,3,4-oxadiazol-2-yl)pyridine
1-(2-methylbenzoyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
2-[1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
5-acetyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2,4-dioxo-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
2-[(2R,3R)-2-hydroxy-3-[(3-methoxypropyl)(methyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]acetic acid
1-{4-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(5-ethyl-2-methylpyrimidin-4-yl)-N-methylpiperidin-3-amine
3-(1,3-benzoxazol-2-yl)-N-(1-propyl-1H-pyrazol-5-yl)piperidine-1-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N,3-diethyl-4-methyl-1H-pyrazole-5-carboxamide
3-{5-[3-(difluoromethoxy)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-indole-6-carboxamide
2-(4-ethylpiperazin-1-yl)-N-[2-(3-methoxyphenyl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one