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1-(2-{1-[(2S)-2-(dimethylamino)-3-phenylpropanoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)propanamide
2-(2-methylphenyl)-5-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}pyrimidine
2-{[(4-chlorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-amino-4-[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
1-{3-oxo-3-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
ethyl 4-[(4-chlorophenyl)methyl]-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylate
2-methoxy-5-oxo-6-[3-(3-oxopiperazin-1-yl)propyl]-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(naphthalene-2-carbonyl)piperidine
2,5-dimethyl-N-(2-methylprop-2-en-1-yl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-(4-fluorophenyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopropane-1-carboxamide
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
6-methoxy-N-[1-(1,3-thiazol-2-yl)propyl]pyrimidin-4-amine
3,8-bis[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-8-[(3-methyl-1H-pyrazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane
4-(4-ethyl-1H-pyrazol-5-yl)-1-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]piperidine
5-benzyl-5-{1-[(9-ethyl-9H-carbazol-3-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
N-methyl-3-phenyl-5-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-3-ylmethyl)benzamide
2-(1H-1,3-benzodiazol-1-yl)-1-[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}acetamide
N-[(1S,2S)-2-(benzyloxy)cyclohexyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-{2-[(dimethylamino)methyl]phenoxy}benzamide
1-(2H-1,3-benzodioxol-5-yl)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]piperidin-4-amine
5-(1-{[(1-cyclohexyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)thiophene-2-carboxamide
2-(2-aminoethyl)-N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]quinazolin-4-amine
1-[7-(2-fluorobenzoyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidine
6-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)pyrimidin-4-ol
1-{2-[5-(2-cyanophenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidine-3-carboxamide
5-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-3-(5-methylfuran-2-yl)-1H-pyrazole
N-methyl-N-[2-(2-{2-[(propan-2-yl)amino]pyrimidin-5-yl}-1H-imidazol-1-yl)ethyl]methanesulfonamide
1-(azepan-1-yl)-3-(3-{[(2-hydroxyethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
5-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(2S,4S)-4-amino-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyrrolidine-2-carboxamide
2-[(1S,5R)-3-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-3-(pyrrolidin-1-ylmethyl)piperidine
2-(dimethyl-1,3-thiazol-5-yl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
1-(oxan-4-yl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
1-(3-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propyl)piperidin-3-ol
4-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N,N-dimethylpiperazine-1-sulfonamide
2-methyl-6-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-6H,7H-[1,3]oxazolo[5,4-d]pyrimidin-7-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-ylmethyl)acetamide
2-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-2-(thiophen-2-ylformamido)propanamide
1-({3-[(5-ethyl-1,3,4-thiadiazol-2-yl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
N-cycloheptyl-N-methyl-2-(oxolan-2-ylmethoxy)acetamide
5-methyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzoxazole
4-{[({3-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]methyl}hepta-1,6-dien-4-ol
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide