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3-{2-[4-(cyclopropylmethyl)piperazin-1-yl]-2-oxoethyl}-4-[(3-fluorophenyl)methyl]piperazin-2-one
N,1-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-S-(4-fluoro-3-methylphenyl)-2-oxoethane-1-sulfonamido
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidine-4-carboxylic acid
2-hydroxy-N-[(3R,4S)-1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-(1-benzothiophene-5-carbonyl)-4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]propan-1-one
N-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(2-methoxyethyl)furan-3-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidine-4-carboxamide
N-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-methyl-1-oxopropan-2-yl}thiophene-2-carboxamide
2-cyclopropyl-9-(3-hydroxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}piperidin-4-amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidine
7-(2-methoxybenzenesulfonyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(2-ethoxypyridin-3-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
ethyl 4-[6-(cyclopent-1-ene-1-carbonyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
ethyl 1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperidine-2-carboxylate
methyl 3-{[1-(4,7-dimethylquinazolin-2-yl)azepan-4-yl]amino}propanoate
(1R,5S,8R)-3-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
7-(2-methylphenyl)-4-[3-(1H-pyrazol-1-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-1,4-diazepan-6-ol
4-({1-[2-(dimethylcarbamoyl)ethyl]pyrrolidin-3-yl}methyl)benzoic acid
3-[2-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]-1,3-oxazinan-2-one
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2-hydroxy-N-methyl-4-(methylsulfanyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]butanamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-propylpyrrolidin-3-yl]-1-(4-methoxyphenyl)cyclopropane-1-carboxamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
5-[(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-{1-[3-(2-methylphenoxy)azetidin-1-yl]-1-oxobutan-2-yl}-2,3-dihydro-1H-isoindol-1-one
3-(4-methoxy-2-methylbenzoyl)-1-(5-methoxyfuran-2-carbonyl)piperidine
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2R,3S,6R)-5-(oxane-4-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(2-hydroxyphenyl)ethyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[2-(propan-2-yl)pyrimidine-4-carbonyl]pyrrolidin-3-yl]methanol
N-ethyl-5-({methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyrimidin-2-amine
3-{2-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
6-(1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)pyrimidin-4-ol
methyl 6-[4-(1H-indol-3-yl)butan-2-yl]-2-(methylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-3-ol
4-hydroxy-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
ethyl 1-(5-methylpyrazine-2-carbonyl)-4-(2-phenylethyl)piperidine-4-carboxylate
1-[3-(2-methylphenoxy)azetidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
3-(3-methoxyquinoxalin-2-yl)-N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]propanamide
2-(3-methoxyphenyl)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
methyl 5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
(1R,3S)-3-methoxy-7-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
methyl 4-{[(2S,4R)-2-[(propan-2-yl)carbamoyl]-4-(pyridin-2-ylsulfanyl)pyrrolidin-1-yl]methyl}benzoate