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4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-(propan-2-yl)-1H-pyrazole
1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
2-[3-(morpholin-4-ylmethyl)phenyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[(5-methylpyrazin-2-yl)methyl]pyrrolidin-2-one
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
6-fluoro-3-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-3,4-dihydroquinazolin-4-one
3-(2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl](pyridin-2-ylmethyl)amine
2-methanesulfonyl-N-{2-[methyl(phenyl)amino]propyl}acetamide
1,5-dimethyl-4-{6-oxo-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
6-(4-methoxyphenyl)-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
(1S,5R)-6-(3,5-difluoropyridine-2-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
2,6-difluoro-3-methyl-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
2-methyl-4-{3-[3-(pyridin-3-yloxy)azetidine-1-carbonyl]phenyl}butan-2-ol
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
2-({[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
5-(1H-imidazol-1-ylmethyl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}furan-2-carboxamide
N-{1-[(4-fluorophenyl)methyl]-7-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
3-benzyl-N-[2-(methylsulfanyl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-ethyl-4-{[methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
1-[5-({[2-(diethylamino)ethyl](ethyl)amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
5-({8-cyclopentyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
N-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]-2-(morpholin-3-yl)acetamide
6-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3-hydroxyphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
N-tert-butyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(1,3,4-thiadiazol-2-yl)urea
[2-(diethylamino)-2-(furan-2-yl)ethyl][(3-fluoro-4-methoxyphenyl)methyl]amine
1-[(4-methoxyphenyl)methyl]-4-[(6-methylquinolin-5-yl)methyl]piperazin-2-one
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]urea
3-({[2-(benzylamino)pyrimidin-5-yl]methyl}(ethyl)amino)-1λ6-thiolane-1,1-dione
N-cyclopropyl-4-{[1-(1-methyl-1H-pyrazol-5-yl)propyl]sulfamoyl}benzamide
(3R,4R)-1-[(6-ethoxypyridin-3-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
(2E)-N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-2-yl)prop-2-enamide
{1-[4-(4-{[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)furan-3-carboxamide
2-{4-[1-(5-methoxyfuran-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-1,4-oxazepan-6-ol
4-[4-(3,4-diethoxyphenyl)-1H-imidazol-2-yl]piperidine
1-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N'-cyclooctyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]butanediamide
5-[(1,3-benzothiazol-2-ylmethyl)(methyl)amino]-1-benzyl-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-chloro-2-(2,2-dimethylmorpholine-4-carbonyl)-3-phenyl-1H-indole
2-(dimethylamino)-2-(4-fluorophenyl)-N-[3-(furan-2-yl)propyl]acetamide
N-[2-(dimethylamino)ethyl]-2-(2-methyl-1H-indol-3-yl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(1-hydroxy-2-methylpropan-2-yl)piperidine-3-carboxamide