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1-{3-oxo-3-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(4-benzylpiperidin-1-yl)-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
4-methyl-1-(2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2-dihydroquinolin-2-one
3-(5-methylfuran-2-yl)-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
6-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-N,N-dimethylpyrazine-2-carboxamide
2-{2-[(6-ethyl-4-methylquinolin-2-yl)amino]ethoxy}ethan-1-ol
5-{[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
methyl (2R,4S)-1-(2,4-difluorobenzenesulfonyl)-4-hydroxypiperidine-2-carboxylate
1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[2-(piperidin-1-yl)ethyl]-1,4-diazepan-5-one
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(3-methoxyphenyl)piperidine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-3-ol
[(3S,5R)-1-[(8-fluoroquinolin-2-yl)methyl]-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
[(4-methoxy-2-methylphenyl)methyl]({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]quinoline-4-carboxylic acid
3-(2-amino-1,3-thiazol-4-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
(2S,4S)-N-ethyl-4-(4-fluoro-3-methoxybenzamido)-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxamide
N-cyclobutyl-3-{[3-(pyridin-2-yl)azetidin-1-yl]sulfonyl}benzamide
1-cyclobutanecarbonyl-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)piperidine-4-carboxamide
N-[2-(4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}morpholin-2-yl)ethyl]acetamide
N-cyclohexyl-N-[(4-fluorophenyl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-{3-[(4-chlorophenyl)sulfanyl]propyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
4-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)pyridine
4-(1H-imidazol-1-yl)-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine-4-carboxylic acid
1-ethyl-N-[(2-methoxyphenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aR,7aS)-1-benzyl-4-(3-hydroxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-4-(morpholin-4-yl)-1-(quinoline-6-carbonyl)pyrrolidin-3-ol
methyl[1-(4-methylpyridin-2-yl)propan-2-yl](pyridin-3-ylmethyl)amine
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-3-sulfamoylthiophene-2-carboxamide
3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(morpholin-4-yl)pyridine-3-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
1-(2-fluorophenyl)-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
N-cyclobutyl-4-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)sulfamoyl}benzamide
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
5-(methoxymethyl)-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
6-methyl-5-{5-[4-methyl-3-(1H-pyrrol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
8-(2-amino-9H-purin-6-yl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]pyrimidin-2-amine
1-[(3,5-difluoro-4-methoxyphenyl)methyl]-N,N-dimethylazepan-4-amine
4-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
1-methyl-1'-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-[(2-methylphenyl)methyl]-4-{[4-(pyridin-2-yl)phenyl]methyl}piperazine
2-{3-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]phenyl}-1H-imidazole
N-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
4-[3-(4-fluorophenoxy)propyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}({2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl})amine
2-methyl-6-(piperidin-4-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrimidin-4-amine
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl]-2-methoxyacetamide