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N-[3-(1H-indol-2-yl)phenyl]-1-(1H-pyrazol-3-ylmethyl)piperidine-3-carboxamide
3-[2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
1-(azocan-1-yl)-3-(5-methoxy-2-{[(3-methoxypropyl)amino]methyl}phenoxy)propan-2-ol
2-{[(3-ethoxyphenyl)methyl](3-methylbut-2-en-1-yl)amino}ethan-1-ol
2-{[4-(3-methyl-1-benzofuran-2-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]oxy}acetic acid
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
(3aS,7aR)-2-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-[4-(5-propyl-1,2-oxazole-3-carbonyl)piperazine-1-carbonyl]morpholine
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
1-[1-(5-chloropyridine-3-carbonyl)piperidin-4-yl]piperidin-4-ol
N-[3-(dimethylamino)propyl]-N-methyl-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-amine
[(3S,7S)-5-(2-amino-6-methylpyrimidin-4-yl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
N-(2-methoxyethyl)-2,4-dimethylpyrimidine-5-carboxamide
N4-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-6-(propan-2-yloxy)pyrimidine-2,4-diamine
methyl 2-{[(4-fluoro-2-methoxyphenyl)methyl]amino}pyridine-4-carboxylate
2-butyl-N-(5-chloro-2-methoxyphenyl)-4-methyl-3-oxopiperazine-1-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-2-methoxy-N-[(3S)-2-oxoazepan-3-yl]acetamide
5-benzyl-5-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-3-(pyridin-3-ylmethyl)imidazolidine-2,4-dione
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-(1,2-oxazolidin-2-ylmethyl)piperidin-2-one
2-(2-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenoxy)ethan-1-ol
N-benzyl{[2-(piperidin-1-ylmethyl)phenyl]amino}sulfonamide
5-[3-(aminomethyl)pyrrolidin-1-yl]-2-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
2-(pyridin-3-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
8-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-1-(3-fluoropyridin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-methanesulfonylpropanamide
N-(4-methyl-1,3-thiazol-2-yl)-5-[1-(1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
(2E)-3-(4-methoxyphenyl)-1-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}prop-2-en-1-one
1-({5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
3-(4-hydroxyphenyl)-N-[2-(pyridin-3-yloxy)propyl]-1H-pyrazole-5-carboxamide
4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]-N-ethylpiperidine-1-carboxamide
2-methyl-4-(5-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}furan-2-yl)but-3-yn-2-ol
1-[(2-methoxyphenyl)methyl]-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazine
N-cyclopentyl-2-(1,3-thiazol-4-yl)-N-(thiophen-3-ylmethyl)acetamide
2-{4-[(6-ethoxyquinolin-2-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
4-{2-cyclohexyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidine
N-methyl-2-[methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]acetamide
2-(2-{1-[2-(pyridin-2-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-cyclopropyl-N-[(4-hydroxyphenyl)methyl]-1H-pyrazole-3-carboxamide
2-({[(2S)-1-hydroxybutan-2-yl]amino}methyl)-6,8-dimethylquinolin-4-ol
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(2,3,6-trifluorophenyl)methyl]amine
ethyl 1-(4-acetylbenzoyl)-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
N-(propan-2-yl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
1-[(2S,4R)-1-benzyl-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-(1-methylpiperidin-4-yl)piperazine
3-(2-methyl-1H-imidazol-1-yl)-1-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}propan-1-one
2-(3-methoxypiperidin-1-yl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridine
4-[(4-methoxyphenyl)methyl]-1-[4-(trifluoromethyl)benzoyl]-1,4-diazepan-5-one
N-{2-[1-(but-2-yn-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}cyclohexanecarboxamide