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2-[(2-chlorophenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]morpholine
2-{4-[3-(2-phenylethyl)piperidin-1-yl]piperidine-1-carbonyl}pyrazine
2-(2,8-dimethylquinoline-3-carbonyl)-2,7-diazaspiro[4.5]decane
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(3,4,5-trimethoxyphenyl)methyl]amine
1-{5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]thiophen-2-yl}ethan-1-one
3-[(3S,4R)-1-benzyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-cyclopentylpropanamide
1-benzyl-4-cyclopropanecarbonyl-1,4-diazepan-6-ol
4-{2-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]ethyl}phenol
7-[2-(3-methoxypropyl)piperidine-1-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
N-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
7-fluoro-3-(morpholin-4-ylmethyl)-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
1-(azepan-1-yl)-3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propan-1-one
2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(pyridin-2-ylmethyl)acetamide
{1-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
9-{[6-(dimethylamino)pyridin-3-yl]methyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-8-(quinoxalin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
4-(2-cyclopropaneamidophenyl)-N,N-dimethylbenzamide
3-[2-(2-hydroxyethoxy)ethyl]-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(3S,4R)-1-[4-methyl-6-(methylsulfanyl)quinolin-2-yl]-4-propylpyrrolidin-3-yl]acetamide
3-(3-fluorophenyl)-N-(3-hydroxy-3-phenylpropyl)-N-methyl-1H-pyrazole-4-carboxamide
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
1-[2-methoxy-5-({[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)morpholine-4-sulfonamide
8-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
N-(1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
3-{[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]methyl}-5-(oxolan-2-yl)-1,2,4-oxadiazole
ethyl 1-cyclopropanecarbonyl-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
1-[4-(1H-pyrazol-3-yl)benzoyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-amine
N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
4-[4-(ethanesulfonyl)piperazin-1-yl]-6-ethyl-2-(pyrrolidin-1-yl)pyrimidine
ethyl 4-{1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carbonyl}piperazine-1-carboxylate
methyl 5-[2-(4-fluorophenyl)piperidin-1-yl]-5-oxopentanoate
3-(propan-2-yl)-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1,2-oxazole-5-carboxamide
6-(4-acetylphenyl)-2-methyl-2,3-dihydropyridazin-3-one
1,1-dioxo-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
1-{1-[4-(hydroxymethyl)pyridine-2-carbonyl]piperidin-4-yl}-3-methylbutan-1-ol
N-[4-(1H-pyrazol-1-yl)butan-2-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-[6-hydroxy-4-(9H-purin-6-yl)-1,4-diazepan-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
3-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-1-[3-(sulfamoylmethyl)phenyl]urea
5-(2,3-dihydro-1-benzofuran-5-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-hydroxy-N-[2-(1-methylpiperidin-3-yl)ethyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[3-cyclopentyl-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
4-[(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)carbamoyl]pyridin-1-ium-1-olate
(3S)-1-[(1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
(1S,5S)-N-(8-chloroquinolin-5-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(1R,3S)-N-(5-chloro-2-methoxyphenyl)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carboxamide