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7-(propan-2-yl)-2-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(4-methyl-2-{4-[1-(morpholin-4-yl)ethyl]phenyl}phenoxy)acetamide
ethyl 2-(1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}piperidin-2-yl)acetate
(1S,5R)-6-[(2-fluoro-4-methoxyphenyl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazin-1-yl]pyridine-3-carbonitrile
(4S)-4-(propan-2-yl)-3-[(2,3,6-trifluorophenyl)methyl]-1,3-oxazolidin-2-one
9-ethyl-4-(2-ethylpyridine-4-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(2-methylfuran-3-carbonyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-acetyl-8-(2-methoxy-5-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
2-(2,3-dihydro-1-benzofuran-7-yl)-2-[4-(pyridin-3-yloxy)piperidin-1-yl]acetic acid
ethyl (2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-propyl-1,2,4-oxadiazol-3-yl)piperidin-3-ol
1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)piperidine-4-carboxylic acid
2-cyclohexyl-1-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethan-1-one
1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-(1H-pyrazol-1-yl)butan-1-one
(5S)-5-[({[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
6-[(4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,3-oxazol-2-yl)methoxy]quinoline
1-(cyclopent-3-ene-1-carbonyl)-4-methanesulfonyl-1,4-diazepane-6-carboxylic acid
4-[({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzene-1-sulfonamide
7-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[(3S,4R)-1-(1H-indole-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
3-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
3-[(3R,4S)-4-(morpholin-4-yl)-1-[(2-phenylethyl)carbamoyl]piperidin-3-yl]propanoic acid
1-{1-[4-(furan-2-yl)benzoyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
N-[(2-ethoxypyridin-3-yl)methyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-1-(3,5-dimethylphenyl)piperazin-2-one
2-{[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]methyl}-6-methylquinolin-4-ol
7-(3-chlorophenyl)-4-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(5-{1-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(3-methoxybenzoyl)piperazine
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[3-(1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decane
3-chloro-4-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[1-(methylsulfanyl)propan-2-yl]piperidine-4-carboxylate
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-2-(2,4,6-trifluorophenyl)ethan-1-one
8-(1-hydroxypropan-2-yl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{5-benzyl-4-[2-(methylsulfanyl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-indole
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(1-methyl-1H-indol-5-yl)methyl]pyrrolidin-3-yl]methanol
(1r,4r)-4-[(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]cyclohexan-1-ol
1-methyl-3-(2-methylpropyl)-5-(2-methylpyrrolidine-1-carbonyl)-1H-pyrazole
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(2-hydroxyphenyl)ethan-1-one
(furan-2-ylmethyl)(prop-2-en-1-yl){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
2-methyl-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-3-[(pyridin-3-ylmethyl)amino]benzamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carboxamide
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
{4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]phenyl}methanol
2-{1-[(4-ethoxyphenyl)methyl]-4-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol