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2-cyclopropanecarbonyl-6-methyl-5-{5-[1-(2-methyl-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[2-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-oxoethyl]pyrrolidin-2-one
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(piperidin-1-yl)butanamide
1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(1S,5R)-6-(2,6-difluoro-3-methoxybenzoyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-amino-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenylpyrimidine-5-carboxamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-6-(methoxymethyl)pyrimidine
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-ethyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
2-[2-({4-butyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1H-pyrrol-1-yl]pyrimidine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
(4S)-3,3,4-trimethyl-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-4-ol
({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)(pyridin-2-ylmethyl)amine
(2S,4R)-4-({[3-(benzyloxy)phenyl]methyl}amino)-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-2-(5-methyl-1H-pyrazol-1-yl)acetamide
2-[5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-(2-methoxyethyl)-4,5-dimethyl-N-(thiophen-2-ylmethyl)thiophene-2-carboxamide
1,6-dimethyl-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-ethyl-4-methyl-1,3-oxazole
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N,N,5-trimethylpyrimidin-4-amine
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)-4-(trifluoromethyl)benzamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)acetamide
N4-[(2-phenyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-(4-ethoxy-2-fluorophenyl)-1-{3-[(5-methylpyridin-2-yl)amino]propyl}urea
3-methyl-2-[1-(1,2-oxazol-5-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-1H-indole
4-methyl-2-[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
3,5-difluoro-2-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
(3aR,6aS)-5-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
{2-[3-(1-methyl-1H-imidazole-2-carbonyl)phenyl]phenyl}methanol
(2E)-N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-N-cyclopentyl-3-(4-methoxyphenyl)prop-2-enamide
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[(3-methylpyridin-2-yl)methyl]amine
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
3-[1-(1-methyl-1H-imidazol-2-yl)butyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
4-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}piperazin-2-one
8-chloro-2-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}quinoline
4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
(2E)-3-(4-methoxyphenyl)-1-{4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}prop-2-en-1-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
1-ethyl-N,N-dimethyl-3-(6-methylquinolin-5-yl)-1H-1,2,4-triazol-5-amine
1-(pyridin-4-ylmethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,4-diazepane
4-[5-({3-[3-(pyridin-4-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,2-oxazol-3-yl]pyridine
(3S,4S)-3-hydroxy-4-(2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)-1λ6-thiolane-1,1-dione
3-[4-(2-fluoro-3-methoxyphenyl)-1H-pyrazol-1-yl]propanamide