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N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(2-hydroxyphenoxy)acetamide
4-[4-(ethanesulfonyl)piperazin-1-yl]-5-ethyl-2-methylpyrimidine
2-[2-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)phenoxy]ethan-1-ol
(4aS,8aR)-6-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
1-methyl-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
1-{1'-[(1R,3S)-3-aminocyclohexanecarbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
4-({2-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)-1,3-thiazol-2-amine
2-[1-({4-[4-(furan-2-carbonyl)piperazin-1-yl]quinazolin-2-yl}methyl)piperidin-2-yl]ethan-1-ol
(3E)-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}hept-3-enoic acid
1-(4-fluorophenyl)-6,6-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-(4-methyl-1,3-thiazol-5-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
2-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]pyridin-3-ol
2-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-4-carbonitrile
7-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
5-cyclopentyl-2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(methylsulfanyl)propan-1-one
4-benzyl-3-ethyl-1-(4-methyl-1,3-oxazole-5-carbonyl)-1,4-diazepan-5-one
1-(2-methyl-4-{[2-(propan-2-yloxy)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
8-{[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
3-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
8-[2-(5-acetylthiophen-3-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-cyclopropyl-6-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrimidin-4-ol
2-{3-[6-amino-5-cyano-4-(4-hydroxyphenyl)pyridin-2-yl]-1H-indol-1-yl}propanoic acid
1-(2-hydroxy-5-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}phenyl)ethan-1-one
1-[2-(4-fluorophenyl)azetidin-1-yl]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propan-1-one
3-cyclohexyl-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-4-carboxamide
N-methyl-N-(2-phenylethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
(2-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}ethyl)dimethylamine
2-(dimethyl-1,2-oxazol-4-yl)-1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
3-{[(cyclohexylmethyl)amino]methyl}-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(thiophen-2-ylmethyl)piperazine
N-ethyl-2,2-dimethyl-4-oxo-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-3,4-dihydro-2H-pyran-6-carboxamide
1-[3-(azepane-1-carbonyl)phenyl]-3-[3-(4-methyl-1H-pyrazol-1-yl)propyl]urea
2-[3-(4-chlorophenyl)-1-propyl-1H-1,2,4-triazol-5-yl]ethan-1-ol
N-cyclobutyl-6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(4-chlorophenyl)-N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]cyclopropane-1-carboxamide
1-(carbamoylmethyl)-N-methyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperidine-3-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
9-(cyclopropylmethyl)-1-methyl-4-(1,3-thiazol-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-3-methylthiophene-2-carboxamide
3-{[2-(2,3-difluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}-N,2-dimethylpropanamide
{3-[4-(4-chlorophenyl)piperazin-1-yl]propyl}diethylamine
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-N-[(3,4,5-trimethoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
N-(2,4-difluorophenyl)-4-(dimethylamino)azepane-1-carboxamide
2-(3-chlorophenyl)-2-hydroxy-N-[2-(2-oxopyrrolidin-1-yl)ethyl]acetamide
2-(4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazin-1-yl)pyrimidine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-phenyl-1-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]piperidine
1-{5-[5-(hydroxymethyl)furan-2-yl]-3-(1H-indol-3-yl)-1H-1,2,4-triazol-1-yl}butan-2-ol