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3-chloro-N-cyclopentyl-4-({1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
5-methyl-5-(3-oxo-3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}propyl)pyrrolidin-2-one
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2H-1,3-benzodioxole-5-carboxamide
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-N-[2-(morpholin-4-yl)ethyl]pyrimidin-2-amine
7-[(2,3-difluorophenyl)methyl]-2-[3-(methylsulfanyl)propyl]-2,7-diazaspiro[4.5]decan-6-one
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(piperidin-4-yl)piperidine
5-(3-fluorophenoxymethyl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
2-methyl-2-[4-(morpholin-4-yl)-2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl]propanoic acid
N-[5-(ethylcarbamoyl)-2-methylphenyl]-4-[2-(pyrrolidin-1-yl)ethyl]piperazine-1-carboxamide
6-methyl-N-propyl-5-[5-(pyrazin-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
1-{4-[2-(2-benzylmorpholin-4-yl)-2-oxoethyl]phenyl}imidazolidin-2-one
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-[(2S)-pyrrolidine-2-carbonyl]piperidine
6-fluoro-N-methyl-N-[(6-methylpyridin-2-yl)methyl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
(2R)-1-{4-[2-oxo-2-(piperidin-1-yl)ethoxy]benzoyl}pyrrolidine-2-carboxamide
2-(4-methylphenyl)-5-[4-(pyridin-2-yl)piperazine-1-carbonyl]pyrimidin-4-ol
(1S,5R)-6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(4aR,8aR)-6-[2-(3-methoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-2-methoxy-2-phenylethan-1-one
5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(4-aminoquinolin-8-yl)benzoic acid
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
methyl[3-(morpholin-4-yl)propyl]{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-({2-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]acetamido}methyl)-4-methylbenzoic acid
1-(3-methylpiperidin-1-yl)-3-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}propan-1-one
N-cyclopropyl-3-[cyclopropyl(1,3-thiazol-2-ylmethyl)sulfamoyl]benzamide
6-[2-(cyclohex-1-en-1-yl)acetyl]-N-[4-(1H-pyrazol-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
5-{1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
4-{2-[1-(oxane-4-carbonyl)piperidin-2-yl]ethyl}phenol
6-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
5-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]pyridin-2-ol
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
(3R,4R)-1-[3-(methoxymethyl)benzoyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[2-(1H-indol-3-yl)ethyl]-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
2-(3-phenylpropyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclopentyl-N-({4-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)ethane-1-sulfonamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
3-[3-cyclopentyl-5-(1-methyl-6-oxo-1,6-dihydropyridazin-3-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]furan-2-carboxamide
8-methyl-2-propyl-N-[2-(1H-pyrrol-1-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(3-methylpyridin-4-yl)-4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
(2S)-2-amino-4-[1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]butanoic acid
N-[(2R,3R)-1'-[2-(cyclohex-1-en-1-yl)acetyl]-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
6-[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carbonyl]-2,3-dihydropyridazin-3-one
N-methyl-5-oxo-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]pyrrolidine-3-carboxamide
9-(3-propyl-1H-pyrazole-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2,2-dimethyl-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)butanamide
1-ethyl-3-(2-methylpropyl)-N-(pyrrolidin-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-{4-[3-(2-phenylethyl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione