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(1R,2R,6S,7S)-4-[1-(4-phenylphenyl)-1H-1,2,3,4-tetrazol-5-yl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-6-methylpyridine-3-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1-(4-methylphenyl)piperazin-2-one
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
5-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}-3-(propan-2-yl)-1,2-oxazole
2,6-diamino-4-(3-chloro-5-fluoro-4-methoxyphenyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
4-(4-methanesulfonylphenyl)-1-[(4-methoxyphenyl)methyl]-1H-pyrazole
(1R,5S)-6-({5-[(3-fluoropyridin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-azabicyclo[3.2.1]octane
2-(3-aminopyrrolidine-1-carbonyl)-6-(2,5-dimethylfuran-3-yl)-7-(3-methylbut-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-3-phenyl-1,2,4-oxadiazole
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-hydroxyphenyl)ethyl]acetamide
4-(2-ethylpyridine-4-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
4-(2H-1,3-benzodioxole-5-carbonyl)-7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-benzyl-3-ethyl-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-5-one
N,4-dimethyl-3-oxo-N-[1-(pyridin-3-yl)propyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(3S,4S)-1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-(4-fluorophenyl)-2-{[3-(1H-pyrazol-1-yl)phenyl]formamido}propanoic acid
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-[(2-methoxyethyl)amino]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
2-{5-[(2-chloro-6-fluorophenyl)methyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-(2-ethyl-1H-imidazol-1-yl)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
6,7-dimethyl-4-({[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]amino}methyl)-2H-chromen-2-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[4-(propan-2-yl)piperazin-1-yl]methyl}piperidin-2-one
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N-ethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-methyl-2-[4-(1-{[(2-methyl-2H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)phenoxy]acetamide
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]propanamide
3-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]propan-1-ol
N-ethyl-2-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]pyridine-4-carboxamide
4-(hydroxymethyl)-4-(oxan-2-ylmethyl)-N-[4-(trifluoromethyl)phenyl]piperidine-1-carboxamide
(2S)-4-methyl-2-({[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]carbamoyl}amino)pentanamide
5-(2-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[methyl(propan-2-yl)amino]methyl}piperidin-2-one
4-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(6-methylpyridazin-3-yl)benzamide
N,N-dimethyl-3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
4-(2-methoxy-6-methylbenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
2-ethyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
5-(2-chlorophenyl)-N-[cyclopropyl(3-methylpyridin-2-yl)methyl]furan-2-carboxamide
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
2-[cyclopentyl(methyl)amino]-1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-fluoro-2-phenylethan-1-one
ethyl 1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-4-[(2-methylphenyl)methyl]piperazin-2-one
1-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-4-[3-(5-methylfuran-2-yl)butyl]piperazine
6-[(diethylamino)methyl]-N-[(5-methylfuran-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(3,4-dichlorophenyl)-4-{imidazo[1,2-a]pyrimidine-2-carbonyl}morpholine
N-methyl-5-[(1,2-oxazol-3-ylmethyl)amino]-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[3-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
1-[4-(3-fluoro-4-methoxyphenyl)phenyl]-2-(morpholin-4-yl)ethan-1-ol