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2-{3-[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-1H-1,3-benzodiazole
{1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
4-({4-[1-(dimethylamino)ethyl]phenyl}methyl)-1-phenylpiperazin-2-one
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4-(2-hydroxypyridine-3-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
5-tert-butyl-4-({2-methyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)furan-2-carboxamide
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3,4-dimethyl-5-sulfamoylbenzamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[(3-chlorophenyl)methyl]-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)propanamide
N-ethyl-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-butyl-4-methyl-6-[4-(pyridin-3-ylmethyl)piperazin-1-yl]pyrimidin-2-amine
2-{[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-methyl-1,3,4-oxadiazole
1-(1H-pyrrole-2-carbonyl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
N-(1H-indol-4-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-[2-(4-methyl-1H-pyrazol-1-yl)phenyl]acetic acid
3-(2-hydroxyethyl)-1-(3-methylbutyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
3-ethyl-5-(2-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,2,4-oxadiazole
N-[2-(furan-2-yl)ethyl]-2-[2-methyl-4-oxo-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-{[5-(furan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-4-methyl-1,3-benzoxazole
6-({2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}amino)pyridine-2-carbonitrile
ethyl 3-benzyl-1-[2-(2-methoxyphenoxy)acetyl]piperidine-3-carboxylate
6-({3-[1-(dimethylamino)ethyl]phenyl}methyl)-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]methylamine
3-(3-methoxyphenyl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
9-(2-ethylpyrimidine-5-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
[7-(3-methoxypyrazin-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
4-(benzyloxy)-1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
4-[(2,4-dimethoxyphenyl)methyl]-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]piperazin-2-one
N-[1-({[2-hydroxy-3-(3-methoxyphenoxy)propyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-phenoxyacetamide
3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-1-(propan-2-yl)piperidine
2-{4-[(3-oxopiperazin-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-({[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[4-({3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)phenyl]imidazolidin-2-one
N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(2-oxopiperidin-1-yl)butanamide
2-(dimethylamino)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-methylphenyl)acetamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(pyrazin-2-yl)piperidine-3-carboxamide
6-{methyl[2-(4-methylpiperazin-1-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
6-(2-chlorophenyl)-2-[4-(piperazin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
2-({[(3R,4R)-1-(5-chloro-2-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-(piperidin-1-ylmethyl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
6-(1-methyl-1H-imidazol-2-yl)-N-(2-phenoxyethyl)pyridazin-3-amine
N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-4-(4-fluorophenyl)-4-hydroxypiperidine-1-carboxamide
N-cyclohexyl-1-methyl-3-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
5-{2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
1-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-[3-(1H-pyrazol-1-yl)phenyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
[(3R,4R)-1-(4-chloro-3-fluorobenzoyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol