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N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-phenyl-1,2-oxazole-4-carboxamide
2-(4-methoxyphenoxy)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
(2S,4R)-4-amino-N,N-diethyl-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)pyrrolidine-2-carboxamide
1-(2-methoxyphenyl)-N-(thiolan-3-yl)-1H-pyrazole-4-carboxamide
6-methyl-N-[2-(morpholin-4-yl)ethyl]-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N'-[(1S)-1-carbamoyl-2-phenylethyl]-N-(2-methylphenyl)propanediamide
(4aR,7aS)-1-propanoyl-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(morpholin-2-yl)-1-[4-(2-phenylethyl)piperidin-1-yl]ethan-1-one
1-cyclopropyl-N-{[4-(morpholin-4-yl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
N-{1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
methyl 4-{[1-(2-methylpropyl)-2,4-dioxo-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
5-cyclobutyl-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1,3,4-oxadiazol-2-amine
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-(5-propyl-1,2-oxazole-4-carbonyl)-1,4-diazepane
N-tert-butyl-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)butanamide
1-{2-oxo-2-[4-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
(1R,7S)-N-methyl-3-[(3-methylphenyl)methyl]-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(3S,4R)-1-(2-methanesulfonylethyl)-4-phenylpyrrolidine-3-carboxylic acid
1-{2-hydroxy-3-[2-methoxy-4-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
N-{1-[1-(1-acetylpiperidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
N-[1-(4-fluorophenyl)piperidin-4-yl]-4-(hydroxymethyl)pyridine-2-carboxamide
methyl 4-{4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazin-1-yl}benzoate
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(1,2-oxazinan-2-yl)propanamide
3-(1-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-1,3-oxazolidin-2-one
{4-[(4-methoxyphenyl)methyl]-1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}methanol
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
(8R,9aS)-8-hydroxy-2-[(1-hydroxycyclohexyl)methyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
4-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}-N,N-dimethylbenzene-1-sulfonamide
1-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}but-3-en-1-one
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
3-[1-(4-methylpyridin-2-yl)-1H-1,3-benzodiazol-2-yl]propan-1-ol
ethyl 1-(2-amino-6-methylpyrimidine-4-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
N-[(2-methoxyphenyl)methyl]-5-methyl-6-(3-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(4-methoxyphenyl)methyl]acetamide
2-{3-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenoxy}acetamide
N-[3-(2-benzyl-3-oxopiperazine-1-carbonyl)phenyl]propanamide
1-methyl-2-[1-(morpholine-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
1-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
4-(2-hydroxy-5-methoxyphenyl)-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)benzonitrile
(2R,6R)-4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-2-(methylsulfanyl)benzamide
3-cyclopropyl-5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
4-chloro-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}benzamide
3-(4-chloro-2-methylbenzoyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
2-(2-hydroxyethyl)-9-[(8-methylquinolin-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[4-(benzyloxy)piperidin-1-yl]-2-(trifluoromethyl)pyrimidine
1-({4-[(E)-2-phenylethenyl]thiophen-2-yl}methyl)piperazine
3-methyl-1-propyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
2-(methoxymethyl)-6-methyl-1-(naphthalen-1-ylmethyl)-3-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
N-[2-(azepan-1-yl)ethyl]-N,1,6-trimethyl-1H-indole-2-carboxamide