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7-hydroxy-6-methyl-4-[(1E)-1-phenylprop-1-en-2-yl]-1,2,3,4-tetrahydroquinolin-2-one
N-cyclopropyl-1-ethyl-N-(1H-indol-5-ylmethyl)piperidine-2-carboxamide
2-hydroxy-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-ethyl-2-methyl-7-oxo-N-(pyridin-4-ylmethyl)-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-(1,2-oxazol-3-ylmethyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
2-{[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl}benzonitrile
3-chloro-4-({1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
1-ethyl-5-methyl-4-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
5-(azepane-1-carbonyl)-N-(1,3-benzothiazol-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(3R,9aR)-8-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{5-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]furan-2-yl}methanol
2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,4-dihydroquinolin-4-one
ethyl 4-(2-phenoxyethyl)-1-[3-(pyridin-3-yl)propanoyl]piperidine-4-carboxylate
5-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N-(2-methylpropyl)furan-2-carboxamide
(2S,4S)-4-amino-1-[(6-chloro-2H-chromen-3-yl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
6-(cyclopropylamino)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-[(4-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}piperidin-1-yl)methyl]pyridine
3-hydroxy-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]propanamide
5-(4-{thieno[3,2-d]pyrimidin-4-yl}phenyl)-1H-pyrazole
{5-[(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-4-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
1-[(3,5-dimethylphenyl)methyl]-4-[2-(methylamino)pyridine-4-carbonyl]piperazin-2-one
[1-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-3-ethylpiperidin-3-yl]methanol
5-[(1-methylpiperidin-4-yl)(pyridin-4-ylmethyl)carbamoyl]-1H-imidazole-4-carboxylic acid
4-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-ethyl-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
5-chloro-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]thiophene-2-carboxamide
1-methyl-3-{2-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}pyrrolidin-2-one
3-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,5-dimethylpyrazine
7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-methyl-N-propyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
1,3-dimethyl-N-[1-(5-methylpyridin-2-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-benzyl-4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperazin-2-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)acetamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-4-methyl-2-oxopentanamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]oxane-2-carboxamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-6-ethylpyrimidin-4-amine
N2-cyclopropyl-N4-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N4-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2-methoxybenzamide
methyl 4-(5-methyl-4-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}-1,3-oxazol-2-yl)benzoate
N-methyl-2-oxo-6-phenyl-N-(quinolin-5-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-(1-cyclohexyl-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazol-3-yl)acetamide
1-(2-{1-[(4-chlorophenyl)methanesulfonyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
5-({[(3-{2-[4-(3,4-dimethoxybenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
N4-cyclopropyl-6-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidine-2,4-diamine
5-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4-propylpyrimidine
2,3,5-trimethyl-7-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}pyrazolo[1,5-a]pyrimidine
2-(2-methoxyethyl)-9-[3-(methylsulfanyl)butyl]-2,9-diazaspiro[5.5]undecan-3-one
6-(2,3-dihydro-1H-inden-1-ylmethyl)-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole