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2-(azepan-1-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide
5-fluoro-2-{1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
(1S,5R)-3-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(3R,4S)-4-(dimethylamino)-1-{[3-(morpholin-4-yl)phenyl]methyl}piperidin-3-yl]propanoic acid
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(cyclopent-2-en-1-yl)ethan-1-one
N-(5-acetamido-2-fluorophenyl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
3-[1-(3-hydroxybutyl)-4-phenyl-1H-imidazol-5-yl]-4-methoxyphenol
4-[(4-fluorophenyl)methyl]-1-(3-methylbut-2-enoyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3-ethyl-5-hydroxyadamantane-1-carboxamide
2-chloro-4-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
N-(1-cyclopentyl-1H-pyrazol-5-yl)-2-[4-(6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]acetamide
[4-({methyl[2-(phenylsulfanyl)ethyl]amino}methyl)oxan-4-yl]methanol
(4aS,8aR)-1-(2-aminoethyl)-6-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
3-methyl-1-{2-oxo-2-[3-(propoxymethyl)pyrrolidin-1-yl]ethyl}-1,2-dihydroquinoxalin-2-one
5-methoxy-2-(3-methyl-1H-pyrazol-1-yl)benzoic acid
(4aS,7aR)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
[(3S,5R)-1-(1-benzothiophene-2-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
8-(oxane-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(8-methoxy-2-methylquinolin-5-yl)-4,6-dimethylpyridine-3-carboxamide
ethyl 1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidine-3-carboxylate
(4aR,7aS)-1-[2-(azepan-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 3-[(3S,4R)-1-[(3-hydroxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
2-[(1S,5R)-6-(2-cyanobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-({1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-3,3,3-trifluoropropanamide
N-(1,4-dithiepan-6-yl)-3,4-dihydro-2H-1-benzopyran-3-amine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
2-[(1S,5R)-6-(2-methoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-[(5-fluoro-2-methylphenyl)methyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxo-2-(thiophen-2-yl)acetamide
6-[4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-1-yl]pyrazine-2-carboxamide
N-cyclopropyl-2-{4-[2-(trifluoromethoxy)phenyl]-1H-1,2,3-triazol-1-yl}acetamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-cyclopentyl-5-oxo-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrrolidine-3-carboxamide
N-benzyl-N-(3-hydroxy-2-methylpropyl)-1-methyl-1H-pyrrole-2-carboxamide
3-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-1,3-oxazolidin-2-one
1-methyl-N-[3-(phenylsulfanyl)propyl]azepane-2-carboxamide
4-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-N-{1-[(methylcarbamoyl)methyl]-1H-pyrazol-4-yl}benzamide
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(pyridin-3-ylmethyl)amine
2-(3-ethylphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
2-[({5-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]furan-2-yl}methyl)sulfanyl]pyrimidine
3-{6-[(2-fluorophenyl)methoxy]-4-[(4-methoxyphenyl)methyl]-3-oxo-1,4-diazepane-1-carbonyl}pyridin-1-ium-1-olate
1-(4-cyclopentyl-6-hydroxy-1,4-diazepan-1-yl)-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
ethyl 5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-methyl-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidine-3-carboxamide
4-methyl-6-(3-{[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrimidin-2-amine
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(oxolan-2-ylmethyl)pyridin-2-amine