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2-methyl-5-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrole-3-carbonitrile
1-[(4aR,8aS)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
5-acetyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
N-({1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-yl}methyl)acetamide
N-{1-[4-(5-methylfuran-2-yl)benzoyl]piperidin-4-yl}methanesulfonamide
2-({imidazo[1,2-a]pyrimidin-2-ylformamido}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-[6-amino-2-(diethylamino)pyrimidin-4-yl]-1-cyclopentylpiperazin-2-one
2-({4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-6-methoxyphenol
(1S,2R)-2-({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl)amino)cyclohexan-1-ol
(2R,3R,6R)-3-(4-fluorophenyl)-N-(furan-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
3-{5-[6-(3-fluorophenyl)pyridin-3-yl]-3-methyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-2-(trifluoromethyl)pyrimidin-4-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[2-(cyclopropylcarbamoyl)ethyl]-N-(3-fluorophenyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-cyclopropyl-3-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]sulfamoyl}benzamide
(3R,4R)-4-(azepan-1-yl)-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-3-ol
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
5-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
N-cyclohexyl-N-[2-(1H-indol-3-yl)ethyl]-3-methyl-1,2-oxazole-5-carboxamide
1-{[2-(2-hydroxyethoxy)phenyl]methyl}-3-(hydroxymethyl)piperidin-3-ol
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
({6-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-methylpyrimidin-4-yl}methyl)dimethylamine
4-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-2,1,3-benzoxadiazole
5-(2,6-dimethylquinoline-4-carbonyl)-N-ethyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{4-[3-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]phenyl}methanol
1-(benzylsulfamoyl)-4-phenylpiperidine-4-carboxylic acid
ethyl 1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-methyl-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-1-phenyl-1H-1,3-benzodiazole-5-carboxamide
N4,6-dimethyl-N2-[1-(2-phenylethyl)piperidin-3-yl]pyrimidine-2,4-diamine
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(pyridin-2-yl)propan-1-one
6-ethyl-2-methyl-4-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]quinoline
1-[(2-chlorophenyl)methyl]-4-(1-ethyl-1H-imidazol-5-yl)-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-methyl-N-(1,2-oxazol-3-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]-N-(1,3-thiazol-2-yl)acetamide
2-cyclopropanecarbonyl-8-(3-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1H-indole
N-[2-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-2-carboxamide
2-{[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
N-cyclopropyl-N-(3-phenylprop-2-yn-1-yl)pyrazolo[1,5-a]pyridine-7-carboxamide
2-(4-{[7-methyl-2-oxo-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-3-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]acetamide
4-[1-(2-{[(4-methoxyphenyl)methyl]carbamoyl}ethyl)piperidin-3-yl]benzoic acid
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2,2,3-trimethylbut-3-en-1-one
5-(3,4-difluorophenoxymethyl)-N-[(1-hydroxycyclohexyl)methyl]-1,2-oxazole-3-carboxamide
1-(1,4-dioxan-2-ylmethyl)-3-[2-(trifluoromethoxy)phenyl]urea
2-(ethylamino)-N-[(4-hydroxyazepan-4-yl)methyl]pyrimidine-5-carboxamide
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-thiazole-4-carboxamide
2-(1-{1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol