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(3S,5R)-1-(3-methoxypropanoyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-[4-(5-phenyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]-1,3-benzoxazole
2-(adamantan-1-yl)-4-hydroxy-N-{[1-(methoxymethyl)cyclopropyl]methyl}pyrimidine-5-carboxamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-[3-(methylamino)propyl]piperidine-3-carboxamide
3-{[1-(4-methylnaphthalene-1-carbonyl)pyrrolidin-3-yl]methyl}benzamide
4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)-N,N-dimethylpiperidine-1-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
1-(cyclohexylmethyl)-N3,N3-dimethyl-N5-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-[4-(furan-2-ylmethoxy)phenyl]urea
1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
N2-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]-N1-(pyridin-3-yl)ethane-1,2-diamine
5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole
2-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(oxolan-2-ylmethyl)acetamide
3-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-1-(2-methoxyethyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
8-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
6-{4-[(3-chloropyridin-4-yl)methyl]piperazin-1-yl}pyrazine-2-carboxamide
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
N-methyl-3-[(4-methylpiperazin-1-yl)sulfonyl]-N-[1-(1,2-oxazol-3-yl)ethyl]-5-phenylbenzamide
1-{[1-(2,5-difluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
N-butyl-4-{2-[(2-methoxyethyl)carbamoyl]ethyl}piperidine-1-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-methyl-1,2,3-thiadiazole-5-carboxamide
1-(4-chloro-1H-pyrazole-3-carbonyl)-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-pyrazol-1-yl)propan-1-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
2-[5-(oxan-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]pyridine
1-(2-aminoethyl)-N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-{[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
(3R,5R)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-(2-methoxyphenyl)-3-{1-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(4aS,7aR)-1-(3,5-dimethylbenzoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-methyl-5-[4-phenyl-1-(prop-2-en-1-yl)-1H-imidazol-5-yl]-1,2-benzoxazole
2-(3-{[8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenoxy)ethan-1-ol
3-{4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2,2-dimethyl-N-(1-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
5-(1-{[5-(2-chlorophenyl)furan-2-yl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(2E)-3-(3-fluorophenyl)-N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}prop-2-enamide
1-(2-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
5-{1-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}-2-methoxypyridine
methyl 3-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)benzoate
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(pyridin-4-yl)propanamide
N-[2-(3-methoxyphenyl)-1-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
1-[2-(1H-imidazol-4-yl)acetyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide