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ethyl 4-(3-phenylpropyl)-1-(1H-pyrazol-3-ylmethyl)piperidine-4-carboxylate
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
N-[2-(azepan-1-yl)ethyl]-N-(propan-2-yl)-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
1-(cyclohexylmethyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-2-(pyridin-3-yl)pyrimidine
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
5-ethyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]pyrimidin-2-amine
1-(2,3-dihydro-1H-inden-2-yl)-4-[3-(1-phenylethyl)-1,2-oxazole-5-carbonyl]-1,4-diazepane
2-(dimethyl-1,2-oxazol-4-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
2-[4-(piperidin-1-ylmethyl)phenyl]-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-{[1-(3,5-dimethylphenyl)cyclopentyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
N-methyl-2-{4-[(3-phenyloxolan-3-yl)methyl]piperazin-1-yl}acetamide
5-[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(cyclohexylmethyl)-5-(oxan-3-ylmethyl)-1H-1,2,4-triazole
(4aR,7aS)-1-(2-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(1,3-thiazol-4-ylmethyl)-decahydroisoquinoline
4-[5-(methoxymethyl)-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
2-(benzyloxy)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
(3R,4S)-4-{4-[4-(1H-pyrazol-3-yl)benzoyl]-1,4-diazepan-1-yl}oxolan-3-ol
7,7-dimethyl-2-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aR,8aR)-2-[(2-aminopyridin-3-yl)methyl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
8-fluoro-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}quinoline-2-carboxamide
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)pyridine-3-carboxylic acid
N-cyclopentyl-N'-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]butanediamide
3-[2-(N-methylmethanesulfonamido)ethyl]-1-(2-methylquinolin-5-yl)urea
(1R,2R,6S,7S)-4-(quinoxaline-5-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
6-methyl-1-{3-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]propyl}-1,2-dihydropyridin-2-one
(1S,2R)-2-[methyl({[1-(propan-2-yl)-1H-imidazol-5-yl]methyl})amino]cyclohexan-1-ol
5-methoxy-9-[3-(1H-pyrazol-1-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecane
2-[(4-methoxyphenyl)methyl]-N-(oxan-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
2,4,5-trimethyl-6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
9-(2-hydroxyethyl)-1-methyl-4-[(2E)-3-phenylprop-2-en-1-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S,4R)-1-[(3-fluorophenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
1-ethyl-4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}pyrrolidin-2-one
1-[2-(azepan-1-yl)-2-oxoethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
[(1,3-dimethylpyrrolidin-3-yl)methyl](methyl){[3-(pyridin-2-ylmethoxy)phenyl]methyl}amine
2-chloro-N-methyl-5-(pyridin-4-yl)benzamide
3-(1-methyl-1H-pyrazol-5-yl)-1-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]propan-1-one
2-{[5-(morpholin-4-ylmethyl)quinolin-8-yl]oxy}pyridine-3-carboxamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-[(3-phenylpropyl)amino]-5-[(propan-2-yl)sulfamoyl]benzamide
N-{1-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-2-(3-methyl-1,2-oxazol-5-yl)acetamide
N-[2-(dimethylsulfamoyl)ethyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
(2S,4S)-N-ethyl-1-(1H-indol-5-ylmethyl)-4-(2-methoxyacetamido)pyrrolidine-2-carboxamide
N-methyl-2-(2-methyl-1H-1,3-benzodiazol-5-yl)-N-[1-(pyridin-3-yl)propyl]acetamide
N-(4-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-4-oxobutyl)acetamide
(1S,4S)-2-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-2-azabicyclo[2.2.1]heptane