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4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-(propan-2-yl)pyrimidine
3-acetamido-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
1-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-3-(trimethyl-1H-pyrazol-4-yl)urea
3-(5-methoxy-2-methylphenyl)-1-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)urea
3-(oxan-4-yl)-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazole
1-(4-methoxyphenyl)-5-methyl-4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-2-one
(1R,5S)-3-[(6-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{[1-(6-methylpyridazin-3-yl)piperidin-4-yl]methyl}benzoic acid
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-3-carboxamide
1-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}imidazolidine-2,4-dione
(3S,4R)-1-cyclohexanecarbonyl-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methyl-N-(1H-pyrazol-5-ylmethyl)benzamide
3-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-1-(thiolan-3-yl)urea
N-(2-hydroxyethyl)-1,4-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-indole-2-carboxamide
1-{[4-(methoxymethyl)piperidin-1-yl]sulfonyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
5-[(2-chloro-6-fluorophenyl)methyl]-1-methyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
1-(morpholin-4-yl)-3-[1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidin-3-yl]propan-1-one
1-ethyl-N-[2-(2-methoxynaphthalen-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-ethyl-5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}pyrimidin-2-amine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-ethyl-N-methyl-5-[(2-phenylethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperazine-2-carboxylic acid
(1R,3S)-3-ethoxy-7-[2-(pyrrolidin-1-yl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
2-{2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
2-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(2S)-2-({5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)-4-(methylsulfanyl)butan-1-ol
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(4-propylpyrimidine-5-carbonyl)piperidin-4-ol
2-({4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
7-(cyclopropylmethyl)-2-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
2-methyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}thieno[2,3-d]pyrimidin-4-amine
1-[4-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-1-methylpiperidine
3-{2-amino-4-methyl-6-[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]pyrimidin-5-yl}propanoic acid
1-(2-methoxyphenyl)-4-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}piperazine
1-(3-methoxypropyl)-2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
1-methyl-3-(propan-2-yl)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
5-cyclobutyl-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1,3,4-oxadiazol-2-amine
N-{2-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]ethyl}acetamide
5-(5-chlorothiophen-2-yl)-1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazole
7-(cyclohexylmethyl)-2-(3-methoxy-4-methylbenzoyl)-2,7-diazaspiro[4.5]decane
5-(dimethoxy-1,3,5-triazin-2-yl)-2-methylquinoline
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[2-(1-methyl-1H-indol-2-yl)pyrimidin-4-yl]pyrrolidin-3-ol
7-(cyclopropylmethyl)-2-{2-[methyl(phenyl)amino]acetyl}-2,7-diazaspiro[4.5]decan-6-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane