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2-(3-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
N-[2-(pyridin-3-yloxy)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-(1-ethylpiperidin-4-yl)ethan-1-one
4-(5-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(3-hydroxy-2,2-dimethylpropyl)amino]methyl}piperidin-2-one
3-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzoic acid
(3S,4R)-3-(dimethylamino)-N-(2-ethoxyphenyl)-4-(4-methylphenyl)pyrrolidine-1-carboxamide
2,3-dimethyl-7-[(3-methyl-1-benzofuran-2-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-ethyl-N,4-dimethyl-1,3-oxazole-5-carboxamide
4-phenyl-1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-one
5-{[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
6-ethyl-2-methoxy-3-{[(oxan-3-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
ethyl 4-[(4-methoxyphenyl)methyl]-1-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]piperidine-4-carboxylate
3-(azepane-1-carbonyl)-N-[(3-methyloxetan-3-yl)methyl]benzene-1-sulfonamide
6-(2-chlorophenyl)-2-(1,4-oxazepane-4-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-methyl-6-[4-(morpholin-4-yl)piperidine-1-carbonyl]thieno[2,3-d]pyrimidin-4-amine
3-(4-methylpiperazine-1-carbonyl)-5-(4-methylpiperidin-1-yl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole
4-[4-({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
2-{4-[4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-6-fluoroquinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
1-(4-methoxyphenyl)-6,6-dimethyl-4-[3-(2-oxopiperidin-1-yl)propanoyl]piperazin-2-one
4,6-dimethyl-1-{2-[5-(5-methylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
2-butyl-8-(6-methyl-2-propylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
{3-[(2-methylphenyl)methyl]-1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl}methanol
4-[6-(3-chloro-2-fluorophenyl)pyridine-3-carbonyl]morpholine
4-ethyl-1-methyl-3-[1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-ethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]thiophene-2-carboxamide
1-({4-methyl-5-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-methylpiperazine-2-carboxylic acid
4-(3-benzyl-1H-pyrazol-5-yl)-1-(1H-pyrrole-2-carbonyl)piperidine
3-(2H-1,3-benzodioxol-5-yl)-5-[(2E)-4-methylpent-2-en-1-yl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-(2-methoxyethyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
5-{5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
N-cyclopentyl-3-(3-hydroxy-1,2-oxazol-5-yl)-N-[(5-methylthiophen-2-yl)methyl]propanamide
(1S,5R)-6-(2-methoxyethyl)-3-(thiophen-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinoline
6-(aminomethyl)-2-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-4-amine
2-[cyclopentyl(methyl)amino]-1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
1-(4-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
4-methoxy-N-methyl-3-(pyridin-3-yl)benzamide
9-(oxane-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-{2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-{[2-(2-fluorophenyl)ethyl]amino}-5-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
[(6-methoxypyridin-3-yl)methyl][(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
8-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-ethyl-4-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-1H-pyrrole-2-carbonitrile
(3R,4S)-1-[6-(piperidin-1-yl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-amine
5-(1-benzyl-4-hydroxypiperidin-4-yl)-N-(4-methoxyphenyl)-1-benzofuran-2-carboxamide