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2-(3,4-dichlorophenyl)-4-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]morpholine
4-(1-methyl-1H-imidazol-2-yl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N,N-dimethyl-4-(4-propylpyrimidine-5-carbonyl)piperazine-1-carboxamide
7-(cyclohexylmethyl)-2-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
1-(cyclopropylmethyl)-5-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4aS,8aR)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-methyl-2-[1-(pyridin-4-yl)piperidin-4-yl]-1H-1,3-benzodiazole
4-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-1-(propan-2-yl)pyrrolidin-2-one
5-methanesulfonyl-2-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]pyrimidin-4-amine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(3-hydroxypropyl)piperidine-3-carboxamide
(2R,3R)-3-amino-1'-(4-methyl-1H-pyrrole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[(5-methylpyrazin-2-yl)methyl]-8-pentyl-2,8-diazaspiro[5.5]undecan-3-one
2-cyclooctyl-4-{4-[4-(4-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
methyl 5-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-cyclohexyl-2-(2,5-dioxoimidazolidin-1-yl)-N-(2-hydroxy-2-phenylethyl)acetamide
(2R)-2-amino-N,4-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pentanamide
2-[2-(carboxymethoxy)phenyl]-1H-1,3-benzodiazole-6-carboxylic acid
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]ethan-1-one
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-2,2-dimethylpropan-1-one
1-[2-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
4-(4-{3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]propanoyl}piperazin-1-yl)benzonitrile
1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(1R,5S,6S)-6-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
methyl 3-(cyclobutylmethoxy)-5-(4-methoxypiperidine-1-carbonyl)benzoate
5-[(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)methyl]-N,N-dimethylfuran-2-carboxamide
1-{4-[({[1-(hydroxymethyl)cyclopentyl]methyl}(methyl)amino)methyl]thiophen-2-yl}ethan-1-one
(2S,4S)-4-amino-1-{1-[(4-methoxyphenyl)amino]cyclohexanecarbonyl}-N-methylpyrrolidine-2-carboxamide
N-(2-methyl-1-oxo-1-{2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}propan-2-yl)thiophene-2-carboxamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
4-(3-methylphenoxy)-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
benzyl(butyl){[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)[1-(pyrimidin-4-yl)ethyl]amine
(4aS,7aR)-1-(2-aminopyridine-4-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4-methoxyphenyl)ethyl]-1-methyl-N-[(1-methylpiperidin-4-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
1-(1H-1,2,3-benzotriazole-5-carbonyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-[(2,5-difluorophenyl)methyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
2-methyl-6-(piperidin-4-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-4-amine
1-{4-[5-(furan-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]phenyl}-1H-pyrazole
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N,1-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-(5-methylthiophen-2-yl)-4-[2-(morpholin-4-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-(cyclobutylmethyl)-2-{[5-(methoxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decane
1'-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-4-[4-(5-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
1-(cyclohexylmethyl)-5-[(3-ethoxypropyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-(3-methyl-3-phenylpiperidin-1-yl)ethan-1-one