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2-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}acetamide
4,6-dimethyl-2-(4-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amino}piperidin-1-yl)pyridine-3-carbonitrile
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
ethyl 4-{[(3S,4R)-3-acetamido-4-propylpyrrolidine-1-carbonyl]amino}benzoate
methyl 6-(1-cyclopentyl-1H-imidazol-2-yl)pyridine-2-carboxylate
1-{4-[2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2,2-dimethylpropan-1-one
N-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}-2-methoxyacetamide
1-[4-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
6-({2-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-1H-imidazol-1-yl}methyl)pyrimidin-4-ol
2-(5-ethyl-1-benzofuran-3-yl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-4-methylbenzamide
4-[3-chloro-4-(prop-2-en-1-yloxy)phenyl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(2-methoxyethyl)piperidine
8-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-[4-(pyrazin-2-yl)piperazine-1-carbonyl]quinoline
1-{2-[({3-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]ethyl}piperidin-2-one
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
N-(prop-2-en-1-yl)-4-(1H-pyrazol-4-yl)benzamide
1-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
2-(4-fluorophenyl)-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
6-fluoro-3-{[1-(2-hydroxyethyl)piperidin-3-yl]methyl}-3,4-dihydroquinazolin-4-one
(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
5-[(1,3-benzothiazol-2-ylmethyl)amino]-1-(cyclohexylmethyl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(2-methoxypyrimidin-5-yl)methyl](2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amine
N-[4-ethoxy-3-(trifluoromethyl)phenyl]-4-(2-methoxyethyl)piperazine-1-carboxamide
6-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(morpholin-4-yl)propan-1-one
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-propanamidobenzamide
2-[4-fluoro-3-(hydroxymethyl)phenyl]-2-{[(2-methoxyphenyl)methyl](methyl)amino}acetic acid
(2S,4S)-4-amino-N-ethyl-1-(5-methylpyridine-3-carbonyl)pyrrolidine-2-carboxamide
1-({3-[(dimethylamino)methyl]phenyl}methyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
(5S)-5-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-2-one
{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-butyl-4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoxaline
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}phenol
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-methyl-N-(1-methylpiperidin-4-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
[3-(2-methoxyethyl)-9-(pyridine-4-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
7-(cyclopropylmethyl)-2-(2-ethylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-ethyl-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-methylpiperidine-3-carboxamide
1-methyl-2-{5-[1-(pyridin-4-ylmethyl)-1H-1,2,3-triazol-4-yl]furan-2-yl}-1H-1,3-benzodiazole
1-(cycloheptylmethyl)-4-phenylpiperazine
2-methyl-N4-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)pyrimidine-4,6-diamine
{4-[(3-chloro-5-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
2-{3-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]phenoxy}propanamide
3-[3-ethyl-3-(hydroxymethyl)piperidine-1-carbonyl]-4-fluorobenzene-1-sulfonamide
3-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-[3-(1H-pyrazol-5-yl)phenyl]urea