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1-(2-methoxyethyl)-8-{[5-(methoxymethyl)furan-2-yl]methyl}-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aS,8aR)-1-(piperidin-4-ylmethyl)-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
ethyl 4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
5-(4-cyclohexylphenyl)-N-[(5-methylpyrazin-2-yl)methyl]-1,2,4-triazin-3-amine
2-({[(3R,4R)-1-(4-chloro-1H-indole-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
[(3R,4R)-1-(3-ethyl-1,2-oxazole-5-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-(3,4-dimethylphenyl)-3-[2-(pyridin-4-yl)-1H-imidazol-1-yl]propanamide
1-{2-[1-(2-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3-benzotriazole
(3S)-1,3-dimethyl-4-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperazin-2-one
ethyl 3-({3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}amino)propanoate
{2-[4-(1-ethoxyethyl)phenyl]pyridin-4-yl}methanol
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-6-sulfonamide
1-{2-[4-benzyl-2-(hydroxymethyl)piperazin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
(4aS,7aR)-1-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-[4-(furan-2-ylmethoxy)phenyl]urea
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(3-phenylpropyl)piperidine-3-carboxamide
(1R,3S,5S)-8-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
1-(cyclopropylmethyl)-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
(1S,5R)-6-(cyclobutylmethyl)-3-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl (1R,3S,3aR,6aS)-5-benzyl-3-(4-hydroxyphenyl)-1-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
{2-[(6-methoxypyrimidin-4-yl)oxy]hex-5-en-1-yl}(methyl)(pyridin-3-ylmethyl)amine
2-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
{4-[(4-methoxyphenyl)methyl]-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl}methanol
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
(3R,4S)-1-(4-chloro-1-methyl-1H-indole-2-carbonyl)-4-(3-methoxyphenyl)pyrrolidin-3-amine
1-(4-{5-[(4-acetylpiperazin-1-yl)methyl]-2-methoxyphenoxy}piperidin-1-yl)-2-[3-(trifluoromethyl)phenyl]ethan-1-one
5-methanesulfonyl-1'-(pyridin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(2,6-dimethoxypyridin-3-yl)-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
6-[4-(1H-pyrazole-4-carbonyl)piperazin-1-yl]-9H-purine
N,N-diethyl-2-({4-[(4-hydroxyphenyl)methyl]-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl}oxy)acetamide
N,6-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(dimethylamino)ethyl]piperidine-3,5-dicarboxamide
1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-3-[(dimethylamino)methyl]piperidin-3-ol
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-2,3-dimethyl-N-(pyridin-3-ylmethyl)-1H-indole-5-carboxamide
N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,3-benzodiazole-5-carboxamide
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxo-N-propylacetamide
3-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(dimethyl-1,3-thiazol-2-yl)methyl]acetamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
3-(pyridin-2-yl)-N-[1-(thiophen-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
3-amino-N-(3-phenylpropyl)-N-(propan-2-yl)benzamide
1-{3-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
1-{6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridin-3-yl}ethan-1-one
(2S,4R)-4-amino-1-(1-benzoylpiperidin-4-yl)-N-methylpyrrolidine-2-carboxamide
N-{1-[1-(4-aminobutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
(1R,3S)-3-({[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}carbamoyl)cyclopentane-1-carboxylic acid
(2S,4R)-4-(dimethylamino)-N-(4-hexylphenyl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide