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N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
7-(cyclobutylmethyl)-2-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-3-methyl-1H-indole-2-carboxamide
2-(3,4-dichlorophenyl)-4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]morpholine
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(6-methoxypyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-[(diethylamino)methyl]-N-methyl-N-[(2-methylphenyl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(dimethylamino)-2-(4-fluorophenyl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-methylpropanamide
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(3-phenyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amine
3-(2H-1,3-benzodioxol-5-yl)-4-methoxybenzamide
2-(1-cyclohexylpiperidin-3-yl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
2-(3-hydroxypropyl)-9-[(4-methoxy-2,3-dimethylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(thian-4-yl)piperazine
3-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-1-ethyl-N,N-dimethyl-1H-1,2,4-triazol-5-amine
(3S,9aR)-3-benzyl-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1S,5R)-3-cyclobutanecarbonyl-6-[2-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-(1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}azetidin-3-yl)-2-methylpiperidine
1-ethyl-3-(morpholine-4-carbonyl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2,7,8-trimethylquinoline-4-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(3-methoxyphenyl)-3-[2-(pyrrolidin-1-yl)propanamido]benzamide
3-[1-(1-benzothiophene-2-carbonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
N-[(3R,4S)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-propylpyrrolidin-3-yl]cyclobutanecarboxamide
(2S,4R)-4-amino-N-(propan-2-yl)-1-[(2,4,5-trimethoxyphenyl)methyl]pyrrolidine-2-carboxamide
1-{1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]piperidin-3-yl}-3-phenylpropan-1-one
6-[(diethylamino)methyl]-N-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-propyl-1H-pyrazole
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]acetamide
5-methyl-3-[1-(1,3-thiazol-2-ylmethyl)pyrrolidin-2-yl]-1,2-oxazole
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(pyridin-3-ylmethyl)propanamide
3,5-dichloro-4-{1-[3-(pyridin-3-yloxy)propyl]-1H-imidazol-2-yl}pyridine
N-ethyl-2-(2-fluorophenoxymethyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(thiophen-3-yl)propan-1-one
(1S,5R)-3-benzyl-6-(4,4,4-trifluorobutyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]benzamide
ethyl({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-1,4-diazepan-5-one
N-[4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-3-phenylpropanamide
1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-4-(1,2-oxazole-3-carbonyl)-1,4-diazepan-6-ol
3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-indazole
1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
(2S,4S)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(2-ethoxyacetamido)-N-ethylpyrrolidine-2-carboxamide
N-benzyl-1-ethyl-N-[(3-methylpyridin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
2-(5-acetylthiophen-3-yl)-N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,2-bis(prop-2-en-1-yl)piperidine