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7-[(2S)-4,4-difluoropyrrolidine-2-carbonyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-3,3-dimethylpiperazin-2-one
7-(cyclopropylmethyl)-2-(3-methyl-1H-indole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,6-dimethoxybenzamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
2-[(3R,4S)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-N,6-dimethylpyrimidin-4-amine
[(3-{[1-(2,5-dimethoxybenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
4-(2,6-dimethylpyridin-3-yl)-2-(1H-pyrrol-2-yl)pyrimidine
5-[6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepane-1-carbonyl]pyridine-2-carbonitrile
5-ethyl-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(2-fluoroethyl)-3-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]sulfamoyl}benzamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
N-(1-cycloheptylpiperidin-3-yl)-1,3-dimethyl-1H-pyrazole-4-sulfonamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-methyl-N-[1-(pyridin-3-yl)propyl]acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methylacetamide
(2S,4S)-4-amino-N-ethyl-1-[3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanoyl]pyrrolidine-2-carboxamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(quinolin-4-yl)-decahydro-1,6-naphthyridin-2-one
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-(pyrimidin-2-yloxy)benzamide
2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-3-carboxylic acid
methyl[(3-methyl-1H-pyrazol-4-yl)methyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
(2S,4S)-4-[2-(dimethyl-1,2-oxazol-4-yl)acetamido]-N-ethyl-1-(oxan-4-yl)pyrrolidine-2-carboxamide
(1-ethyl-5-{2-methylthieno[3,2-d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
9-[2-(propan-2-yl)pyrimidin-4-yl]-2H,3H,6H,7H,8H,9H-[1,4]dioxino[2,3-g]quinolin-7-one
4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperazine-1-sulfonamide
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-(2,2,6,6-tetramethylpiperidin-4-yl)ethan-1-one
(2R)-2-[5-(5-fluoro-3-methyl-1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
2-[5-(2,4-dimethoxyphenyl)-3-(pyridin-2-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
[(3-{2-[4-(2,3-dimethyl-1H-indole-7-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
1'-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-4-ylmethyl)acetamide
5-chloro-2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1,3-benzoxazole
methyl({[1-(morpholin-4-yl)cyclohexyl]methyl}){pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amine
2-(3-methoxypropyl)-9-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(oxolan-2-ylmethyl)-5-phenyl-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
4-(benzylamino)-1-[(4-fluorophenyl)methyl]pyrrolidin-2-one
ethyl 1-ethyl-5-(pyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-fluoro-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
2-[(2-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}phenyl)amino]acetic acid
2-methoxy-N-{4-[4-(1H-pyrazol-5-yl)phenyl]phenyl}acetamide
N-ethyl-5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}pyrimidin-2-amine
5-acetyl-N,2,4-trimethyl-N-[(3-methylpyridin-2-yl)methyl]-1H-pyrrole-3-carboxamide
2-(4-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}piperidin-1-yl)pyrimidine
3,5-dimethyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-indole-2-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(5-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(4-ethenylphenyl)-2-(ethoxymethyl)pyrrolidine-1-carboxamide