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1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
ethyl 4-{methyl[(3-methylthiophen-2-yl)methyl]amino}piperidine-1-carboxylate
6-fluoro-2-({1-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-1,3-benzodiazole
N-ethyl-2-(methylamino)-N-[(2E)-3-phenylprop-2-en-1-yl]pyridine-3-carboxamide
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)amine
1-{[1-(propoxycarbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-(azepan-1-yl)-3-[3-({[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
5-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-6-(methoxymethyl)pyrimidine
3-chloro-5-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
5-[2-(cyclopentylamino)pyrimidin-4-yl]-2-ethoxybenzoic acid
3-[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]propane-1,2-diol
(2S,4S)-1-benzyl-4-[(cyclohexylmethyl)amino]-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
N-ethyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
2-{4-[4-(4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine
1-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-(4-fluorophenyl)morpholin-4-yl]propan-1-one
8-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-1-oxa-8-azaspiro[4.6]undecane
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-phenylethan-1-one
N-[(3S,4R)-1-[2-(2-methyl-1H-indol-3-yl)acetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
5-methyl-1-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-(4-methylpent-3-en-1-yl)piperidin-2-one
3-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)-4-(3-methylbutyl)piperazin-2-one
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
(1S,5R)-3-(2,5-dimethylfuran-3-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-[(2,2-dimethylpropanamido)methyl]benzoate
2-({2-[1-(3-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pyridin-4-ylmethyl)quinoline-2-carboxamide
methyl 2-[(2-benzyl-1-methyl-5-propanamido-1H-1,3-benzodiazol-7-yl)formamido]acetate
3-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
3,5-dimethyl-2-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1H-indole
methyl (2S,4S)-4-(3-fluorobenzamido)-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxylate
4-(1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
N-({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)-N-methyloxan-4-amine
4-cyclobutaneamido-N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
6-[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyridine-3-carboxamide
5-(4-fluorophenyl)-N-(oxan-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
N-(1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
N-[(2,6-difluorophenyl)methyl]-4-(1,3-thiazol-2-yl)morpholine-2-carboxamide
dimethyl[3-({5-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyridin-2-yl}oxy)propyl]amine
4-{[1-(oxolane-3-carbonyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-4-methylpiperidine
3-(4-hydroxyphenyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide
N-[(3-methoxyphenyl)methyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(2-fluorophenyl)methyl]-3-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
5-{[(3-chlorophenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-methyl-5-{1-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazol-3-yl}-N-[(3,4,5-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide