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1-(2,5-dimethoxyphenyl)-3-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}urea
(4aR,7aS)-1-ethyl-4-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aS,6aS)-2-[(2-chloro-4-fluorophenyl)methyl]-5-cyclohexyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(5-methyl-1,2,4-oxadiazol-3-yl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-7-{[(3-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
methyl 4-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-4-oxobutanoate
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide
4-(3-methylphenoxy)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
4-[(4-ethoxyphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 1-(5-acetylthiophene-3-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
N-(1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-5,6,7,8-tetrahydroquinoline-3-carboxamide
[(3S,4S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(hydroxymethyl)pyrrolidin-3-yl]methanol
4-[(3-methoxypyrrolidin-1-yl)methyl]-1-methyl-3-phenyl-1H-pyrazole
6-(1,2,3,4-tetrahydroisoquinolin-5-yl)-1,3-benzothiazol-2-amine
1-(furan-2-ylmethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
N-[(1-phenylcyclopentyl)methyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-[1-(3-methoxypropyl)pyrrolidin-3-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(2S,4S)-4-[2-(carbamoylamino)acetamido]-N-ethyl-1-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
2-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]-N,N-dimethylethane-1-sulfonamide
6-[(diethylamino)methyl]-N-(2-oxopiperidin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
6-methyl-5-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(carbamoylmethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]piperidine-4-carboxamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
ethyl 4-{[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]amino}piperidine-1-carboxylate
9-[2-(ethylamino)pyrimidine-5-carbonyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-tert-butylbenzenesulfonyl)-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
5-methyl-3-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-indole-2-carboxylic acid
5-cyclopropanecarbonyl-1'-(pyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-methoxy-N-[(1-methylpiperidin-3-yl)methyl]-5-(propan-2-yl)benzene-1-sulfonamide
N-methyl-3-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)piperidin-2-one
1-[3-({[2-(2-fluorophenyl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-{2-[2-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
4-({4-methyl-5-[1-(pyridin-4-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
9-(5-fluoropentyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(4-phenylphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-fluorophenyl)methyl]piperazin-2-one
{5-fluoro-7-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
N-butyl-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-[4-(piperidine-1-carbonyl)pyridin-2-yl]benzoic acid
(4aS,7aR)-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
methyl 4-(3-{2-[(5-chloro-2-methoxyphenyl)carbamoyl]ethyl}piperidin-1-yl)-4-oxobutanoate
(2S,4S)-4-amino-1-(3,4-dihydro-2H-1,5-benzodioxepine-7-sulfonyl)-N-methylpyrrolidine-2-carboxamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
6-chloro-2-{2-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one