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[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl](methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N,N,2-trimethyl-7-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(3,4-dimethylphenyl)-1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]piperidin-3-amine
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
3,5-dichloro-N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N,4-dimethylbenzamide
2-{3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]phenoxy}acetamide
8-(2,2-dimethylpropyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,4R)-4-hydroxy-N,1-dimethyl-N-[(3-methylthiophen-2-yl)methyl]piperidine-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
4-(6-aminopyridine-3-carbonyl)-1-cyclopentylpiperazin-2-one
9-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-methoxy-1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
3-[2-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}amino)phenyl]-N-methylpropanamide
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)[(3-methylpyridin-2-yl)methyl]amine
2-amino-N-[5-carbamoyl-2-(3-methylpiperidin-1-yl)phenyl]-6-methylpyrimidine-4-carboxamide
N-{5-[(1R,5R)-3-azabicyclo[3.3.1]nonan-3-ylmethyl]pyrimidin-2-yl}benzenesulfonamide
3-{2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl}pyridine
1-(cyclohexylmethyl)-3-hydroxy-3-[(4-hydroxypiperidin-1-yl)methyl]piperidin-2-one
(3aR,6aR)-N-[2-(2,3-dimethoxyphenyl)ethyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-ethyl-N-(2-fluoro-5-methanesulfonamidophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
8-butanoyl-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-ethyl-2-methylpyrimidin-4-amine
1-benzyl-5-(pyridine-2-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-2-yl]pyridine
2-(3-fluorophenoxymethyl)-N-[1-(2-methylphenyl)cyclopropyl]-1,3-oxazole-4-carboxamide
8-[(4-fluoro-3-methylphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
9-(6-cyclopropylpyrimidin-4-yl)-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1-cyclopentylpiperazin-2-one
N-(4-{5-[(2-methoxypyrimidin-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)acetamide
5-{4-[(3-methoxypyrrolidin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
({3-[(dimethylamino)methyl]phenyl}methyl)(methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
2-[3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenyl]-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(pyridin-3-ylmethyl)piperidin-3-ol
(3S,9aR)-8-(4-chlorobenzoyl)-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(1H-imidazol-1-yl)-N-[(2-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]propanamide
3-[4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]benzonitrile
4-methyl-6-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-3-yl)pyrimidine
1-[(2,6-difluorophenyl)methyl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-(3-hydroxy-2,2-dimethylpropyl)-2-methyl-1-benzofuran-5-carboxamide
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(4-propylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(3R,4R)-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
2-(5-chlorothiophen-2-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazole
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(4aS,8aR)-1-(3-hydroxypropyl)-6-(2-methyl-5-propylpyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
N-ethyl-2-(4-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}piperazin-1-yl)acetamide
2-amino-3-ethyl-N-[2-(1H-indol-3-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine