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dimethyl(3-{[5-(3-methylpyridin-4-yl)pyridin-2-yl]oxy}propyl)amine
3-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indole
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(4-{[1-(1-methylpiperidine-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
2-{1-[(3-acetyl-2,4,6-trimethylphenyl)methyl]piperidin-4-yl}-N-methylacetamide
1-(1,4-diazepan-1-yl)-3-(pyridin-4-yl)propan-1-one
1-{1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}piperidin-3-ol
2-(2,5-dimethylphenyl)-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)acetamide
9-(4-methoxy-3,5-dimethylbenzoyl)-1,4,9-triazaspiro[5.5]undecan-5-one
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]butanamide
2-hydroxy-3-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
4-(4-fluorophenyl)-2-(thiomorpholin-4-ylmethyl)phenol
N-(2-hydroxypropyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
4-(3-chloro-4-methylbenzoyl)-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-6-(2-methoxyphenyl)-N-methylpyridazin-3-amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
2-({2-[(dimethylamino)methyl]phenyl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
5-methyl-4-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1-(2-methylphenyl)piperazin-2-one
(4aS,8aR)-6-(ethanesulfonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(4-methyl-1H-pyrazol-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}propanamide
2-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
7-[4-(1H-pyrazol-1-yl)benzenesulfonyl]-2,7-diazaspiro[4.5]decane
(3S,4S)-1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N,N-diethyl-1-[5-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl]pyrrolidin-3-amine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(dimethyl-1,3-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(3-chlorophenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(2-ethoxyphenyl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)acetamide
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-cycloheptyl-2-[(3R,4S)-3-acetamido-4-propylpyrrolidin-1-yl]acetamide
1-methyl-3-phenyl-8-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,8-diazaspiro[4.5]decane
(3R,4S)-1-(7-fluoro-2-methylquinoline-4-carbonyl)-4-phenylpyrrolidin-3-amine
7-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[(3-chloro-4,5-dimethoxyphenyl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-[(4-fluorophenyl)methyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1-[4-({[2-(1H-indol-1-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
[(3-methoxyphenyl)methyl](prop-2-en-1-yl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
3-acetyl-N-[2-(4-fluorophenyl)ethyl]-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-(2-ethylphenyl)-2-[2-(pyridin-2-yl)acetamido]benzamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-(2-methoxyethoxy)phenyl]azetidine-1-carboxamide
{1-[(6-chloro-2H-chromen-3-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
2-(1-cyclohexyl-4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
N-benzyl{[3-(4-methylpiperazine-1-carbonyl)phenyl]amino}sulfonamide
(3R,9aR)-3-benzyl-8-(2,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-(2,3-dihydro-1H-inden-2-yl)-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
2,6,8-trimethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
(4S)-3-{2-[3-(3-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
1-cyclopropyl-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrrolidin-2-one
6-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-7-methylpyrazolo[1,5-a]pyrimidine
5-cyclopropanecarbonyl-1'-(thiophen-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]