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2-(3-fluorophenyl)-2-{[3-(4H-1,2,4-triazol-4-yl)phenyl]formamido}acetic acid
(3S,4R)-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-(2-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)pyridine
2,2-dimethyl-N-[2-(6-oxo-2-phenyl-1,6-dihydropyrimidin-4-yl)ethyl]-1-(thiophen-2-yl)cyclopropane-1-carboxamide
5-[1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-N-(pyridin-4-yl)thiophene-2-carboxamide
3-{3-[(2R,6S)-2,6-dimethylpiperidin-1-yl]propanoyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
(3aS,6aS)-2-benzyl-5-[3-(pyridin-4-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3R,4R)-1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-4-ethylpiperidine-3,4-diol
[(2,3-difluorophenyl)methyl][2-(1H-imidazol-1-yl)ethyl]methylamine
1-{3-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
2-{4-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]phenoxy}acetamide
methyl 4-{[4-(2-phenylethoxy)phenyl]methyl}piperazine-1-carboxylate
(3R,5R)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
(3R,5S)-N-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
3-[4-(dimethylamino)azepane-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
N-methyl-4-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
(3S,4S)-1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)urea
2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
2-(3-methoxypropyl)-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
6-{[(4-hydroxy-1-methylpiperidin-4-yl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
9-(5-chloropyridine-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2,3-dimethyl-6-[3-(1-methylpiperidin-3-yl)propanoyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-hydroxy-2-phenyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-[1-(4-fluorophenyl)piperidin-4-yl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(3S,4R)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-5-[2-(4-methylbenzenesulfonyl)ethyl]-1H-1,2,4-triazole
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-(pyridin-2-ylmethyl)cyclohexanamine
(3aR,6aS)-1-oxo-5-[(4-phenoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-chlorophenyl)-N-[2-(dimethylamino)ethyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(1-ethyl-1H-indazol-3-yl)-2-[4-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
5-methyl-3-[(4-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H-1,2,3-triazol-1-yl)methyl]-1,2,4-oxadiazole
5-methyl-N-[2-(3-methylpyridin-2-yl)ethyl]-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4-(2-phenoxyethyl)piperazine
2-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-3-ol
2-[4-(piperidin-1-ylmethyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
4-[4-(1H-pyrazol-4-yl)butanoyl]piperazine-2-carboxylic acid
4-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazin-1-yl}-2-methyl-5-propylpyrimidine
2-[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]pyridine-3-carboxamide
8-[(2S)-2-amino-3-hydroxypropanoyl]-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(dimethylamino)ethyl]-3-methoxy-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)propanamide
4-ethyl-6-[4-(4-methoxyphenoxymethyl)piperidin-1-yl]pyrimidine
{2-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[2-(dimethylsulfamoyl)ethyl]-2-(2-methyl-1H-indol-3-yl)acetamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-ethoxyphenyl)methyl]piperidin-3-yl}propanamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-propoxypropanamide
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrazole-3-carbonyl)piperidine